日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Pharmacological inhibition of the Janus Kinases enhances ASCL1 protein stability and transcriptional activity.

Janus激酶的药理学抑制可增强ASCL1蛋白的稳定性和转录活性

Hanspal Maya A, Presland Jeremy, Shkura Kirill, Veiga Martina Koeva, Gillotin Sébastien

Discovery of 5-Amino-N-(1H-pyrazol-4-yl)pyrazolo[1,5-a]pyrimidine-3-carboxamide Inhibitors of IRAK4

发现 5-氨基-N-(1H-吡唑-4-基)吡唑并[1,5-a]嘧啶-3-甲酰胺类 IRAK4 抑制剂

Lim, Jongwon; Altman, Michael D; Baker, James; Brubaker, Jason D; Chen, Hongmin; Chen, Yiping; Fischmann, Thierry; Gibeau, Craig; Kleinschek, Melanie A; Leccese, Erica; Lesburg, Charles; Maclean, John K F; Moy, Lily Y; Mulrooney, Erin F; Presland, Jeremy; Rakhilina, Larissa; Smith, Graham F; Steinhuebel, Dietrich; Yang, Ruojing