日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

TMIC-62. Astrocyte-expressed FASN as a novel candidate drug target for glioblastoma

TMIC-62. 星形胶质细胞表达的FASN作为胶质母细胞瘤的新型候选药物靶点

Van Doorn, C E; Tyree, J B; Jaramillo, A A; Gómez Soria, I; Finneran, Dylan; Jackman, Briana G; Desjarlais, Taylor; Morgan, Dave; Gordon, Marcia N; Kumari, Namrata; Sodders, Maggie; Marathi, Archana; Olsen, Abby; Cho, Kei Kwangwook; Bertherat, Féodora; Carlyle, Becky C; Bengoa‐Vergniory, Nora; Cowley, Sally A; Wade‐Martins, Richard; Carmichael, James Eric; Liu, Martha; Xu, TianMeng; Tuduri, Pola S; Ding, Michelle; Manseau, Frédéric S; Williams, Sylvain; da Silva Mansano, Naira; Wray, Susan; Girijala, Veena; Farias, Antolin Serrano; Suvarnapathaki, Sanika; Traversa, Benito; Aude, Carlos Andres; Torroella, Jordina Rincon; Yi, Li; Massai, Francesco; Moussaud, Simon; Iyer, Preeti; Fitzek, Martina; Preston, Marian; Gaetani, Massimiliano; Schmierer, Bernhard; Gustavsson, Anna-Lena; Smith, Dave; Davis, Andrew; Mega, Alessandro; Östman, Arne

Redirecting raltitrexed from cancer cell thymidylate synthase to Mycobacterium tuberculosis phosphopantetheinyl transferase.

将 raltitrexed 从癌细胞胸苷酸合成酶重定向到结核分枝杆菌磷酸泛酰巯基转移酶

Singh Amrita, Ottavi Samantha, Krieger Inna, Planck Kyle, Perkowski Andrew, Kaneko Takushi, Davis Andrew M, Suh Christine, Zhang David, Goullieux Laurent, Alex Alexander, Roubert Christine, Gardner Mark, Preston Marian, Smith Dave M, Ling Yan, Roberts Julia, Cautain Bastien, Upton Anna, Cooper Christopher B, Serbina Natalya, Tanvir Zaid, Mosior John, Ouerfelli Ouathek, Yang Guangli, Gold Ben S, Rhee Kyu Y, Sacchettini James C, Fotouhi Nader, Aubé Jeffrey, Nathan Carl

Discovery of a novel allosteric inhibitor-binding site in ERK5: comparison with the canonical kinase hinge ATP-binding site

ERK5中一种新型变构抑制剂结合位点的发现:与经典激酶铰链区ATP结合位点的比较

Chen, Hongming; Tucker, Julie; Wang, Xiaotao; Gavine, Paul R; Phillips, Chris; Augustin, Martin A; Schreiner, Patrick; Steinbacher, Stefan; Preston, Marian; Ogg, Derek