日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Development of pyrazolo[1,5-a]pyrimidine based macrocyclic kinase inhibitors targeting AAK1.

开发以吡唑并[1,5-a]嘧啶为基础的大环激酶抑制剂,靶向AAK1。

Mensing Theresa E, Kurz Christian G, Amrhein Jennifer A, Ehret Theresa A L, Preuss Franziska, Mathea Sebastian, Karim Marwah, Tran Do Hoang Nhu, Kadlecova Zuzana, Tolvanen Tuomas A, Martinez-Molina Daniel, Müller Susanne, Einav Shirit, Knapp Stefan, Hanke Thomas

Structural Aspects of LIMK Regulation and Pharmacology

LIMK调控和药理学的结构方面

Chatterjee, Deep; Preuss, Franziska; Dederer, Verena; Knapp, Stefan; Mathea, Sebastian

Lessons from LIMK1 enzymology and their impact on inhibitor design.

从 LIMK1 酶学中汲取的经验教训及其对抑制剂设计的影响

Salah Eidarus, Chatterjee Deep, Beltrami Alessandra, Tumber Anthony, Preuss Franziska, Canning Peter, Chaikuad Apirat, Knaus Petra, Knapp Stefan, Bullock Alex N, Mathea Sebastian