Development of pyrazolo[1,5-a]pyrimidine based macrocyclic kinase inhibitors targeting AAK1.
开发以吡唑并[1,5-a]嘧啶为基础的大环激酶抑制剂,靶向AAK1。
期刊:European Journal of Medicinal Chemistry
影响因子:5.9
doi:10.1016/j.ejmech.2025.118076
Mensing Theresa E, Kurz Christian G, Amrhein Jennifer A, Ehret Theresa A L, Preuss Franziska, Mathea Sebastian, Karim Marwah, Tran Do Hoang Nhu, Kadlecova Zuzana, Tolvanen Tuomas A, Martinez-Molina Daniel, Müller Susanne, Einav Shirit, Knapp Stefan, Hanke Thomas