Click-to-lead design of a picomolar ABA receptor antagonist with potent activity in vivo
利用点击先导化合物设计法合成了一种皮摩尔级ABA受体拮抗剂,该拮抗剂在体内具有强效活性。
期刊:Proceedings of the National Academy of Sciences of the United States of America
影响因子:9.1
doi:10.1073/pnas.2108281118
Vaidya, Aditya S; Peterson, Francis C; Eckhardt, James; Xing, Zenan; Park, Sang-Youl; Dejonghe, Wim; Takeuchi, Jun; Pri-Tal, Oded; Faria, Julianna; Elzinga, Dezi; Volkman, Brian F; Todoroki, Yasushi; Mosquna, Assaf; Okamoto, Masanori; Cutler, Sean R