日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Dimethoxybenzohomoadamantane-based soluble epoxide hydrolase inhibitors: in vivo efficacy in a murine model of chemotherapy-induced neuropathic pain

基于二甲氧基苯并高金刚烷的可溶性环氧化物水解酶抑制剂:在化疗诱导神经性疼痛小鼠模型中的体内疗效

Codony, Sandra; Jora, Beatrice; Santos-Caballero, Miriam; Qiu, Qiongju; Calvó-Tusell, Carla; Escriche, Celia; Turcu, Andreea L; Prischi, Filippo; Bartra, Clara; Val, Cristina; Morisseau, Christophe; Pérez, Belén; Bertran-Mostazo, Andrea; Osuna, Sílvia; Corpas, Rubén; Griñán-Ferré, Christian; Galdeano, Carles; Loza, M Isabel; Pallàs, Mercè; Sanfeliu, Coral; Hammock, Bruce D; Brea, José; Feixas, Ferran; Conte, Maria R; Cobos, Enrique J; Vázquez, Santiago

Enhanced identification of small molecules binding to hnRNPA1 via cryptic pockets mapping coupled with X-ray fragment screening

通过隐蔽口袋定位结合X射线片段筛选,增强对与hnRNPA1结合的小分子的鉴定。

Dunnett, Louise; Das, Sayan; Venditti, Vincenzo; Prischi, Filippo

DrugSynthMC: An Atom-Based Generation of Drug-like Molecules with Monte Carlo Search

DrugSynthMC:一种基于原子的药物分子生成方法,利用蒙特卡罗搜索进行研究。

Roucairol, Milo; Georgiou, Alexios; Cazenave, Tristan; Prischi, Filippo; Pardo, Olivier E

Perspective: Structure determination of protein-ligand complexes at room temperature using X-ray diffraction approaches

展望:利用X射线衍射方法在室温下测定蛋白质-配体复合物的结构

Hough, Michael A; Prischi, Filippo; Worrall, Jonathan A R

Functionally distinct mutations within AcrB underpin antibiotic resistance in different lifestyles.

AcrB 中功能不同的突变是不同生活方式下抗生素耐药性的根本原因

Trampari Eleftheria, Prischi Filippo, Vargiu Attilio V, Abi-Assaf Justin, Bavro Vassiliy N, Webber Mark A

Repurposed floxacins targeting RSK4 prevent chemoresistance and metastasis in lung and bladder cancer

靶向RSK4的新型氟沙星类药物可预防肺癌和膀胱癌的化疗耐药性和转移。

Chrysostomou, Stelios; Roy, Rajat; Prischi, Filippo; Thamlikitkul, Lucksamon; Chapman, Kathryn L; Mufti, Uwais; Peach, Robert; Ding, Laifeng; Hancock, David; Moore, Christopher; Molina-Arcas, Miriam; Mauri, Francesco; Pinato, David J; Abrahams, Joel M; Ottaviani, Silvia; Castellano, Leandro; Giamas, Georgios; Pascoe, Jennifer; Moonamale, Devmini; Pirrie, Sarah; Gaunt, Claire; Billingham, Lucinda; Steven, Neil M; Cullen, Michael; Hrouda, David; Winkler, Mathias; Post, John; Cohen, Philip; Salpeter, Seth J; Bar, Vered; Zundelevich, Adi; Golan, Shay; Leibovici, Dan; Lara, Romain; Klug, David R; Yaliraki, Sophia N; Barahona, Mauricio; Wang, Yulan; Downward, Julian; Skehel, J Mark; Ali, Maruf M U; Seckl, Michael J; Pardo, Olivier E

The role of the p90 ribosomal S6 kinase family in prostate cancer progression and therapy resistance

p90核糖体S6激酶家族在前列腺癌进展和治疗耐药性中的作用

Cronin, Ryan; Brooke, Greg N; Prischi, Filippo

The Role of Ribosomal Protein S6 Kinases in Plant Homeostasis

核糖体蛋白S6激酶在植物体内平衡中的作用

Obomighie, Irabonosi; Lapenas, Kestutis; Murphy, Billy E; Bowles, Alexander M C; Bechtold, Ulrike; Prischi, Filippo

Machine learning application for development of a data-driven predictive model able to investigate quality of life scores in a rare disease

用于开发数据驱动预测模型的机器学习应用程序,该模型能够研究罕见病患者的生活质量评分。

Spiga, Ottavia; Cicaloni, Vittoria; Fiorini, Cosimo; Trezza, Alfonso; Visibelli, Anna; Millucci, Lia; Bernardini, Giulia; Bernini, Andrea; Marzocchi, Barbara; Braconi, Daniela; Prischi, Filippo; Santucci, Annalisa

Cytosine methylation at CpCpG sites triggers accumulation of non-CpG methylation in gene bodies

CpCpG位点的胞嘧啶甲基化会引发基因体内非CpG甲基化的积累。

Zabet, Nicolae Radu; Catoni, Marco; Prischi, Filippo; Paszkowski, Jerzy