日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Consecutive Day HSP90 Inhibitor Administration Improves Efficacy in Murine Models of KIT-Driven Malignancies and Canine Mast Cell Tumors

连续两天给予HSP90抑制剂可提高KIT驱动的恶性肿瘤小鼠模型和犬肥大细胞瘤的疗效

London, Cheryl A; Acquaviva, Jaime; Smith, Donald L; Sequeira, Manuel; Ogawa, Luisa Shin; Gardner, Heather L; Bernabe, Louis Feo; Bear, Misty D; Bechtel, Sandra A; Proia, David A

Ganetespib, an HSP90 inhibitor, kills Epstein-Barr virus (EBV)-infected B and T cells and reduces the percentage of EBV-infected cells in the blood

Ganetespib是一种HSP90抑制剂,它能杀死感染了EB病毒(EBV)的B细胞和T细胞,并降低血液中EBV感染细胞的百分比。

Shatzer, Amber; Ali, Mir A; Chavez, Mayra; Dowdell, Kennichi; Lee, Min-Jung; Tomita, Yusuke; El-Hariry, Iman; Trepel, Jane B; Proia, David A; Cohen, Jeffrey I

Repeated PD-1/PD-L1 monoclonal antibody administration induces fatal xenogeneic hypersensitivity reactions in a murine model of breast cancer

在乳腺癌小鼠模型中,重复注射PD-1/PD-L1单克隆抗体可诱发致命的异种超敏反应。

Mall, Christine; Sckisel, Gail D; Proia, David A; Mirsoian, Annie; Grossenbacher, Steven K; Pai, Chien-Chun Steven; Chen, Mingyi; Monjazeb, Arta M; Kelly, Karen; Blazar, Bruce R; Murphy, William J

STA-8666, a novel HSP90 inhibitor/SN-38 drug conjugate, causes complete tumor regression in preclinical mouse models of pediatric sarcoma

STA-8666 是一种新型 HSP90 抑制剂/SN-38 药物偶联物,可在儿童肉瘤的临床前小鼠模型中引起肿瘤完全消退。

Heske, Christine M; Mendoza, Arnulfo; Edessa, Leah D; Baumgart, Joshua T; Lee, Sunmin; Trepel, Jane; Proia, David A; Neckers, Len; Helman, Lee J

Radioresistant human lung adenocarcinoma cells that survived multiple fractions of ionizing radiation are sensitive to HSP90 inhibition.

能够耐受多次电离辐射的抗辐射人类肺腺癌细胞对 HSP90 抑制剂敏感

Gomez-Casal Roberto, Epperly Michael W, Wang Hong, Proia David A, Greenberger Joel S, Levina Vera

Ganetespib, a novel Hsp90 inhibitor in patients with KRAS mutated and wild type, refractory metastatic colorectal cancer

Ganetespib 是一种新型 Hsp90 抑制剂,用于治疗 KRAS 突变型和野生型难治性转移性结直肠癌患者。

Cercek, Andrea; Shia, Jinru; Gollub, Marc; Chou, Joanne F; Capanu, Marinela; Raasch, Pamela; Reidy-Lagunes, Diane; Proia, David A; Vakiani, Efsevia; Solit, David B; Saltz, Leonard B

Targeted inhibition of Hsp90 by ganetespib is effective across a broad spectrum of breast cancer subtypes

ganetespib 对 Hsp90 的靶向抑制作用对多种乳腺癌亚型均有效。

Friedland, Julie C; Smith, Donald L; Sang, Jim; Acquaviva, Jaime; He, Suqin; Zhang, Chaohua; Proia, David A

Targeted inhibition of the molecular chaperone Hsp90 overcomes ALK inhibitor resistance in non-small cell lung cancer

靶向抑制分子伴侣Hsp90可克服非小细胞肺癌中的ALK抑制剂耐药性

Sang, Jim; Acquaviva, Jaime; Friedland, Julie C; Smith, Donald L; Sequeira, Manuel; Zhang, Chaohua; Jiang, Qin; Xue, Liquan; Lovly, Christine M; Jimenez, John-Paul; Shaw, Alice T; Doebele, Robert C; He, Suqin; Bates, Richard C; Camidge, D Ross; Morris, Stephan W; El-Hariry, Iman; Proia, David A

Synergistic activity of the Hsp90 inhibitor ganetespib with taxanes in non-small cell lung cancer models

Hsp90抑制剂ganetespib与紫杉烷类药物在非小细胞肺癌模型中的协同作用

Proia, David A; Sang, Jim; He, Suqin; Smith, Donald L; Sequeira, Manuel; Zhang, Chaohua; Liu, Yuan; Ye, Shuxia; Zhou, Dan; Blackman, Ronald K; Foley, Kevin P; Koya, Keizo; Wada, Yumiko