日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Preclinical characterization and clinical translation of pharmacodynamic markers for MK-5890: a human CD27 activating antibody for cancer immunotherapy

MK-5890(一种用于癌症免疫治疗的人源CD27激活抗体)的药效学标志物的临床前表征和临床转化

Lars Guelen ,Thierry O Fischmann ,Jerelyn Wong ,Smita Mauze ,Marco Guadagnoli ,Nikolina Bąbała ,Jozef Wagenaars ,Veronica Juan ,David Rosen ,Winnie Prosise ,Maurice Habraken ,Imke Lodewijks ,Danling Gu ,Judith Stammen-Vogelzangs ,Ying Yu ,Jeanne Baker ,David Lutje Hulsik ,Lilian Driessen-Engels ,Dan Malashock ,Joost Kreijtz ,Astrid Bertens ,Evert de Vries ,Astrid Bovens ,Arne Bramer ,Yiwei Zhang ,Richard Wnek ,Sean Troth ,Elliot Chartash ,Konstantin Dobrenkov ,Svetlana Sadekova ,Andrea van Elsas ,Jason K Cheung ,Laurence Fayadat-Dilman ,Jannie Borst ,Amy M Beebe ,Hans Van Eenennaam

Pembrolizumab microgravity crystallization experimentation

帕博利珠单抗微重力结晶实验

Reichert, Paul; Prosise, Winifred; Fischmann, Thierry O; Scapin, Giovanna; Narasimhan, Chakravarthy; Spinale, April; Polniak, Ray; Yang, Xiaoyu; Walsh, Erika; Patel, Daya; Benjamin, Wendy; Welch, Johnathan; Simmons, Denarra; Strickland, Corey

Structure of the insulin receptor-insulin complex by single-particle cryo-EM analysis

通过单粒子低温电子显微镜分析胰岛素受体-胰岛素复合物的结构

Giovanna Scapin, Venkata P Dandey, Zhening Zhang, Winifred Prosise, Alan Hruza, Theresa Kelly, Todd Mayhood, Corey Strickland, Clinton S Potter, Bridget Carragher

A novel storage system for cryoEM samples

一种新型的冷冻电镜样品存储系统

Scapin, Giovanna; Prosise, Winifred W; Wismer, Michael K; Strickland, Corey

Discovery of Novel 3,3-Disubstituted Piperidines as Orally Bioavailable, Potent, and Efficacious HDM2-p53 Inhibitors

发现新型3,3-二取代哌啶类化合物作为口服生物利用度高、效力强、疗效显著的HDM2-p53抑制剂

Bogen, Stéphane L; Pan, Weidong; Gibeau, Craig R; Lahue, Brian R; Ma, Yao; Nair, Latha G; Seigel, Elise; Shipps, Gerald W Jr; Tian, Yuan; Wang, Yaolin; Lin, Yinghui; Liu, Ming; Liu, Suxing; Mirza, Asra; Wang, Xiaoying; Lipari, Philip; Seidel-Dugan, Cynthia; Hicklin, Daniel J; Bishop, W Robert; Rindgen, Diane; Nomeir, Amin; Prosise, Winifred; Reichert, Paul; Scapin, Giovanna; Strickland, Corey; Doll, Ronald J

Joint angles and angular velocities and relevance of eigenvectors during prehension in the monkey

猴子抓握过程中关节角度、角速度及特征向量的相关性

Prosise, Jodi F; Hendrix, Claudia M; Ebner, Timothy J

Discovery of a Potent, Injectable Inhibitor of Aurora Kinases Based on the Imidazo-[1,2-a]-Pyrazine Core

基于咪唑并[1,2-a]吡嗪核心结构,发现了一种强效的、可注射的Aurora激酶抑制剂

Yu, Tao; Tagat, Jayaram R; Kerekes, Angela D; Doll, Ronald J; Zhang, Yonglian; Xiao, Yushi; Esposite, Sara; Belanger, David B; Curran, Patrick J; Mandal, Amit K; Siddiqui, M Arshad; Shih, Neng-Yang; Basso, Andrea D; Liu, Ming; Gray, Kimberly; Tevar, Seema; Jones, Jennifer; Lee, Suining; Liang, Lianzhu; Ponery, Samad; Smith, Elizabeth B; Hruza, Alan; Voigt, Johannes; Ramanathan, Lata; Prosise, Winifred; Hu, Mengwei

Key steps in the structure-based optimization of the hepatitis C virus NS3/4A protease inhibitor SCH503034

丙型肝炎病毒NS3/4A蛋白酶抑制剂SCH503034的结构优化关键步骤

Madison, Vincent; Prongay, Andrew J; Guo, Zhuyan; Yao, Nanhua; Pichardo, John; Fischmann, Thierry; Strickland, Corey; Myers, Joseph Jr; Weber, Patricia C; Beyer, Brian M; Ingram, Richard; Hong, Zhi; Prosise, Winifred W; Ramanathan, Lata; Taremi, S Shane; Yarosh-Tomaine, Taisa; Zhang, Rumin; Senior, Mary; Yang, Rong Sheng; Malcolm, Bruce; Arasappan, Ashok; Bennett, Frank; Bogen, Stephane L; Chen, Kevin; Jao, Edwin; Liu, Yi Tsung; Lovey, Raymond G; Saksena, Anil K; Venkatraman, Srikanth; Girijavallabhan, Viyyoor; Njoroge, F George

Construction, expression, and characterization of a novel fully activated recombinant single-chain hepatitis C virus protease

构建、表达和表征一种新型全活化重组单链丙型肝炎病毒蛋白酶

Taremi, S S; Beyer, B; Maher, M; Yao, N; Prosise, W; Weber, P C; Malcolm, B A