日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Design, Synthesis, Biological Evaluation, and In Silico Studies of Novel Multitarget Cinnamic Acid Hybrids

新型多靶点肉桂酸杂合物的设计、合成、生物学评价和计算机模拟研究

Tsopka, Ioanna-Chrysoula; Pontiki, Eleni; Sigala, Ioanna; Nikolakaki, Eleni; Prousis, Kyriakos C; Hadjipavlou-Litina, Dimitra

Novel Multi-Target Agents Based on the Privileged Structure of 4-Hydroxy-2-quinolinone

基于4-羟基-2-喹啉酮特殊结构的新型多靶点药物

Kostopoulou, Ioanna; Tzani, Andromachi; Chronaki, Konstantina; Prousis, Kyriakos C; Pontiki, Eleni; Hadjiplavlou-Litina, Dimitra; Detsi, Anastasia

A quest for the stereo-electronic requirements for selective agonism for the neurotrophin receptors TrkA and TrkB in 17-spirocyclic-dehydroepiandrosterone derivatives

探索 17-螺环脱氢表雄酮衍生物中神经营养因子受体 TrkA 和 TrkB 选择性激动的立体电子要求

Daniele Narducci, Despoina Charou, Thanasis Rogdakis, Ioanna Zota, Vivi Bafiti, Maria Zervou, Theodora Katsila, Achille Gravanis, Kyriakos C Prousis, Ioannis Charalampopoulos, Theodora Calogeropoulou

Development and Biological Characterization of a Novel Selective TrkA Agonist with Neuroprotective Properties against Amyloid Toxicity

新型选择性TrkA激动剂的开发和生物学表征及其对淀粉样蛋白毒性的神经保护作用

Thanasis Rogdakis ,Despoina Charou ,Alessia Latorrata ,Eleni Papadimitriou ,Alexandros Tsengenes ,Christina Athanasiou ,Marianna Papadopoulou ,Constantina Chalikiopoulou ,Theodora Katsila ,Isbaal Ramos ,Kyriakos C Prousis ,Rebecca C Wade ,Kyriaki Sidiropoulou ,Theodora Calogeropoulou ,Achille Gravanis ,Ioannis Charalampopoulos

Synthesis and Antifouling Activity Evaluation of Analogs of Bromosphaerol, a Brominated Diterpene Isolated from the Red Alga Sphaerococcus coronopifolius

从红藻冠状球藻(Sphaerococcus coronopifolius)中分离得到的溴代二萜化合物溴球醇类似物的合成及防污活性评价

Prousis, Kyriakos C; Kikionis, Stefanos; Ioannou, Efstathia; Morgana, Silvia; Faimali, Marco; Piazza, Veronica; Calogeropoulou, Theodora; Roussis, Vassilios

Accelerating Drug Discovery Efforts for Trypanosomatidic Infections Using an Integrated Transnational Academic Drug Discovery Platform

利用综合跨国学术药物研发平台加速锥虫病药物研发工作

Carolina B Moraes, Gesa Witt, Maria Kuzikov, Bernhard Ellinger, Theodora Calogeropoulou, Kyriakos C Prousis, Stefano Mangani, Flavio Di Pisa, Giacomo Landi, Lucia Dello Iacono, Cecilia Pozzi, Lucio H Freitas-Junior, Bruno Dos Santos Pascoalino, Claudia P Bertolacini, Birte Behrens, Oliver Keminer, J

BNN27, a 17-Spiroepoxy Steroid Derivative, Interacts With and Activates p75 Neurotrophin Receptor, Rescuing Cerebellar Granule Neurons from Apoptosis

BNN27,一种17-螺环氧类固醇衍生物,与p75神经营养因子受体相互作用并激活该受体,从而挽救小脑颗粒神经元免于凋亡。

Iosif Pediaditakis ,Alexandra Kourgiantaki ,Kyriakos C Prousis ,Constantinos Potamitis ,Kleanthis P Xanthopoulos ,Maria Zervou ,Theodora Calogeropoulou ,Ioannis Charalampopoulos ,Achille Gravanis

Identification of Novel Chemical Scaffolds Inhibiting Trypanothione Synthetase from Pathogenic Trypanosomatids

从致病性锥虫中鉴定抑制锥虫硫合成酶的新型化学骨架

Benítez, Diego; Medeiros, Andrea; Fiestas, Lucía; Panozzo-Zenere, Esteban A; Maiwald, Franziska; Prousis, Kyriakos C; Roussaki, Marina; Calogeropoulou, Theodora; Detsi, Anastasia; Jaeger, Timo; Šarlauskas, Jonas; Peterlin Mašič, Lucíja; Kunick, Conrad; Labadie, Guillermo R; Flohé, Leopold; Comini, Marcelo A

Synthesis and Crystal Structure Characterization of Zinc (II) Tetronic Acid Complexes

锌(II)四氢萘酸配合物的合成及晶体结构表征

Prousis, K C; Athanasellis, G; Stefanou, V; Matiadis, D; Kokalari, E; Igglessi-Markopoulou, O; McKee, V; Markopoulos, J

Synthesis of “Acetylene-Expanded” Tridentate Ligands

“乙炔扩展”三齿配体的合成

Matiadis, Dimitris; Prousis, Kyriakos C; Igglessi-Markopoulou, Olga; Holmes, Brian T; Pennington, William T; Hanks, TW