日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Synthesis and Characterization of Photoswitchable Covalent Ligands for the β(2)-Adrenoceptor

β(2)-肾上腺素受体光开关共价配体的合成与表征

Wirth, Ulrike; Neu, Eduard; Provasi, Davide; Feustel, Steffen; Schmidt, Maximilian F; Hübner, Harald; Weikert, Dorothée; Filizola, Marta; König, Burkhard; Gmeiner, Peter

Structural basis for saxitoxin congener binding and neutralization by anuran saxiphilins.

无尾目石房蛤毒素结合蛋白对石房蛤毒素同系物结合和中和的结构基础

Zakrzewska Sandra, Nixon Samantha A, Chen Zhou, Hajare Holly S, Park Elizabeth R, Mulcahy John V, Arlinghaus Kandis M, Neu Eduard, Konovalov Kirill, Provasi Davide, Leighfield Tod A, Filizola Marta, Du Bois J, Minor Daniel L Jr

Geometry-Driven Control of Linear and Nonlinear Optical Responses in p‑Nitroaniline: Insights into Structure-Property Relationships and Thermal Robustness

几何结构驱动的对硝基苯胺线性和非线性光学响应控制:结构-性质关系和热稳定性的深入研究

Manzoni, Vinicius; Gester, Rodrigo M; da Cunha, Antônio R; Pagola, Gabriel I; Quinteiro Rosen, Guillermo F; Provasi, Patricio F

Synthesis, Biotransformation, Characterization, and DFT Study of Organic Azachalcone Dyes and Secondary Metabolites with Biological and Conformation Dependence of Dipolar-Octupolar NLO Responses

有机氮杂查尔酮染料及其次级代谢产物的合成、生物转化、表征和DFT研究,以及偶极-八极非线性光学响应的生物学和构象依赖性

Ribeiro, Victoria L; Dos Santos, Neidy S S; de Oliveira, Raira V S; Carvalho, Joselina A; Garcia, Viviane V; Brito-Junior, Hartmann J S; Usfinit, Willibrodus; Pinheiro, Mayra; Fill, Taicia; Gester, Rodrigo; Provasi, Patricio F; Canuto, Sylvio; Bitencourt, Heriberto R; Marinho, Patricia S B; Marinho, Andrey M R

Fine-Tuned Deep Transfer Learning Models for Large Screenings of Safer Drugs Targeting Class A GPCRs

用于大规模筛选靶向A类GPCR的更安全药物的精细化深度迁移学习模型

Provasi, Davide; Filizola, Marta

Coping and quality of life of parents of children with achondroplasia-a narrative review

软骨发育不全患儿父母的应对方式和生活质量——一项叙述性综述

Adedeji, Adekunle; Witt, Stefanie; Innig, Florian; Alves, Inês; Provasi, Chiara; Sessa, Marco; Mohnike, Klaus; Quitmann, Julia

BOLD-GPCRs: A Transformer-Powered App for Predicting Ligand Bioactivity and Mutational Effects Across Class A GPCRs

BOLD-GPCRs:一款基于Transformer的预测A类GPCR配体生物活性和突变效应的应用程序

Provasi, Davide; Konovalov, Kirill; Riina, Nicholas; Cullen, Olivia; Filizola, Marta

Structural and dynamic studies uncover a distinct allosteric modulatory site at the μ-opioid receptor

结构和动力学研究揭示了μ-阿片受体上一个独特的变构调节位点。

Zhang, Haonan; Konovalov, Kirill; Parpounas, Alexandra K; Provasi, Davide; Yang, Shifan; Abraham, Alejandro; Warren, Audrey L; Zilberg, Gregory; Wang, Suri; Filizola, Marta; Wacker, Daniel

Elucidating the molecular logic of a metabotropic glutamate receptor heterodimer

阐明代谢型谷氨酸受体异二聚体的分子逻辑

Lin, Xin; Provasi, Davide; Niswender, Colleen M; Asher, Wesley B; Javitch, Jonathan A

Structural insights into the unexpected agonism of tetracyclic antidepressants at serotonin receptors 5-HT1eR and 5-HT1FR

四环抗抑郁药对血清素受体 5-HT1eR 和 5-HT1FR 的意外激动作用的结构洞察

Gregory Zilberg, Alexandra K Parpounas, Audrey L Warren, Bianca Fiorillo, Davide Provasi, Marta Filizola, Daniel Wacker