日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Investigation of the molecular characteristics of bisindole inhibitors as HIV-1 glycoprotein-41 fusion inhibitors

对双吲哚抑制剂作为HIV-1糖蛋白-41融合抑制剂的分子特性进行研究

Zhou, Guangyan; Chu, Shidong; Nemati, Ariana; Huang, Chunsheng; Snyder, Beth A; Ptak, Roger G; Gochin, Miriam

An analog of camptothecin inactive against Topoisomerase I is broadly neutralizing of HIV-1 through inhibition of Vif-dependent APOBEC3G degradation

一种对拓扑异构酶I无活性的喜树碱类似物,可通过抑制Vif依赖的APOBEC3G降解,广泛中和HIV-1病毒。

Bennett, Ryan P; Stewart, Ryan A; Hogan, Priscilla A; Ptak, Roger G; Mankowski, Marie K; Hartman, Tracy L; Buckheit, Robert W Jr; Snyder, Beth A; Salter, Jason D; Morales, Guillermo A; Smith, Harold C

HIV-1, human interaction database: current status and new features

HIV-1 人类相互作用数据库:现状及新增功能

Ako-Adjei, Danso; Fu, William; Wallin, Craig; Katz, Kenneth S; Song, Guangfeng; Darji, Dakshesh; Brister, J Rodney; Ptak, Roger G; Pruitt, Kim D

Structure-activity relationships of a novel capsid targeted inhibitor of HIV-1 replication

一种新型衣壳靶向HIV-1复制抑制剂的构效关系

Kortagere, Sandhya; Xu, Jimmy P; Mankowski, Marie K; Ptak, Roger G; Cocklin, Simon

Discovery and optimization of novel small-molecule HIV-1 entry inhibitors using field-based virtual screening and bioisosteric replacement

利用基于场的虚拟筛选和生物等排置换法发现和优化新型小分子HIV-1进入抑制剂

Tuyishime, Marina; Danish, Matt; Princiotto, Amy; Mankowski, Marie K; Lawrence, Rae; Lombart, Henry-Georges; Esikov, Kirill; Berniac, Joel; Liang, Kuang; Ji, Jingjing; Ptak, Roger G; Madani, Navid; Cocklin, Simon

Dimeric RNA recognition regulates HIV-1 genome packaging

二聚体RNA识别调控HIV-1基因组包装

Nikolaitchik, Olga A; Dilley, Kari A; Fu, William; Gorelick, Robert J; Tai, S-H Sheldon; Soheilian, Ferri; Ptak, Roger G; Nagashima, Kunio; Pathak, Vinay K; Hu, Wei-Shau

Identification of a small-molecule inhibitor of HIV-1 assembly that targets the phosphatidylinositol (4,5)-bisphosphate binding site of the HIV-1 matrix protein

鉴定出一种靶向HIV-1基质蛋白磷脂酰肌醇(4,5)-二磷酸结合位点的HIV-1组装小分子抑制剂

Zentner, Isaac; Sierra, Luz-Jeannette; Fraser, Ayesha K; Maciunas, Lina; Mankowski, Marie K; Vinnik, Andrei; Fedichev, Peter; Ptak, Roger G; Martín-García, Julio; Cocklin, Simon

Discovery of a small-molecule antiviral targeting the HIV-1 matrix protein

发现一种靶向HIV-1基质蛋白的小分子抗病毒药物

Zentner, Isaac; Sierra, Luz-Jeannette; Maciunas, Lina; Vinnik, Andrei; Fedichev, Peter; Mankowski, Marie K; Ptak, Roger G; Martín-García, Julio; Cocklin, Simon

Development of real-time PCR array for simultaneous detection of eight human blood-borne viral pathogens

开发用于同时检测八种人类血液传播病毒病原体的实时PCR芯片

Pripuzova, Natalia; Wang, Richard; Tsai, Shien; Li, Bingjie; Hung, Guo-Chiuan; Ptak, Roger G; Lo, Shyh-Ching

Mechanisms of human immunodeficiency virus type 2 RNA packaging: efficient trans packaging and selection of RNA copackaging partners

人类免疫缺陷病毒2型RNA包装机制:高效反式包装和RNA共包装伴侣的选择

Ni, Na; Nikolaitchik, Olga A; Dilley, Kari A; Chen, Jianbo; Galli, Andrea; Fu, William; Prasad, V V S P; Ptak, Roger G; Pathak, Vinay K; Hu, Wei-Shau