日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Novel Class of Chikungunya Virus Small Molecule Inhibitors That Targets the Viral Capping Machinery

一类新型的基孔肯雅病毒小分子抑制剂,靶向病毒加帽机制

Abdelnabi, Rana; Kovacikova, Kristina; Moesslacher, Julia; Donckers, Kim; Battisti, Verena; Leyssen, Pieter; Langer, Thierry; Puerstinger, Gerhard; Quérat, Gilles; Li, Changqing; Decroly, Etienne; Tas, Ali; Marchand, Arnaud; Chaltin, Patrick; Coutard, Bruno; van Hemert, Martijn; Neyts, Johan; Delang, Leen

Structure Elucidation of Coxsackievirus A16 in Complex with GPP3 Informs a Systematic Review of Highly Potent Capsid Binders to Enteroviruses.

柯萨奇病毒 A16 与 GPP3 复合物的结构解析为高效肠道病毒衣壳结合剂的系统评价提供了依据

De Colibus Luigi, Wang Xiangxi, Tijsma Aloys, Neyts Johan, Spyrou John A B, Ren Jingshan, Grimes Jonathan M, Puerstinger Gerhard, Leyssen Pieter, Fry Elizabeth E, Rao Zihe, Stuart David I

More-powerful virus inhibitors from structure-based analysis of HEV71 capsid-binding molecules

基于HEV71衣壳结合分子的结构分析,发现了更强效的病毒抑制剂

De Colibus, Luigi; Wang, Xiangxi; Spyrou, John A B; Kelly, James; Ren, Jingshan; Grimes, Jonathan; Puerstinger, Gerhard; Stonehouse, Nicola; Walter, Thomas S; Hu, Zhongyu; Wang, Junzhi; Li, Xuemei; Peng, Wei; Rowlands, David; Fry, Elizabeth E; Rao, Zihe; Stuart, David I

The imidazopyrrolopyridine analogue AG110 is a novel, highly selective inhibitor of pestiviruses that targets the viral RNA-dependent RNA polymerase at a hot spot for inhibition of viral replication

咪唑并吡咯并吡啶类似物AG110是一种新型的高选择性瘟病毒抑制剂,它靶向病毒RNA依赖性RNA聚合酶的关键位点,从而抑制病毒复制。

Paeshuyse, Jan; Chezal, Jean-Michel; Froeyen, Matheus; Leyssen, Pieter; Dutartre, Hélène; Vrancken, Robert; Canard, Bruno; Letellier, Carine; Li, Tong; Mittendorfer, Harald; Koenen, Frank; Kerkhofs, Pierre; De Clercq, Erik; Herdewijn, Piet; Puerstinger, Gerhard; Gueiffier, Alain; Chavignon, Olivier; Teulade, Jean-Claude; Neyts, Johan

A novel, highly selective inhibitor of pestivirus replication that targets the viral RNA-dependent RNA polymerase

一种新型的、高选择性的瘟病毒复制抑制剂,靶向病毒RNA依赖性RNA聚合酶。

Paeshuyse, Jan; Leyssen, Pieter; Mabery, Eric; Boddeker, Nina; Vrancken, Robert; Froeyen, Matheus; Ansari, Israrul H; Dutartre, Hélène; Rozenski, Jef; Gil, Laura H V G; Letellier, Carine; Lanford, Robert; Canard, Bruno; Koenen, Frank; Kerkhofs, Pierre; Donis, Ruben O; Herdewijn, Piet; Watson, Julia; De Clercq, Erik; Puerstinger, Gerhard; Neyts, Johan