Design of Potent and Selective Covalent Inhibitors of Bruton's Tyrosine Kinase Targeting an Inactive Conformation
针对布鲁顿酪氨酸激酶非活性构象设计高效选择性共价抑制剂
期刊:ACS Medicinal Chemistry Letters
影响因子:4
doi:10.1021/acsmedchemlett.9b00317
Pulz, Robert; Angst, Daniela; Dawson, Janet; Gessier, Francois; Gutmann, Sascha; Hersperger, Rene; Hinniger, Alexandra; Janser, Philipp; Koch, Guido; Revesz, Laszlo; Vulpetti, Anna; Waelchli, Rudolf; Zimmerlin, Alfred; Cenni, Bruno