日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Unraveling the Potential of Amino‑, Acylamino‑, and Ureido-Substituted 3H‑1,2-Benzoxaphosphepine 2‑Oxides toward Nanomolar Inhibitors of Tumor-Associated Carbonic Anhydrases IX and XII

揭示氨基、酰氨基和脲基取代的3H-1,2-苯并氧杂磷杂环庚烷2-氧化物作为肿瘤相关碳酸酐酶IX和XII纳摩尔级抑制剂的潜力

Balašova, Anastasija; Pustenko, Aleksandrs; Angeli, Andrea; Andreucci, Elena; Biagioni, Alessio; Nocentini, Alessio; Carta, Fabrizio; Supuran, Claudiu T; Žalubovskis, Raivis

The antibiotic furagin and its derivatives are isoform-selective human carbonic anhydrase inhibitors

抗生素呋喃妥因及其衍生物是具有同工酶选择性的人类碳酸酐酶抑制剂。

Pustenko, Aleksandrs; Nocentini, Alessio; Gratteri, Paola; Bonardi, Alessandro; Vozny, Igor; Žalubovskis, Raivis; Supuran, Claudiu T