Unraveling the Potential of Amino‑, Acylamino‑, and Ureido-Substituted 3H‑1,2-Benzoxaphosphepine 2‑Oxides toward Nanomolar Inhibitors of Tumor-Associated Carbonic Anhydrases IX and XII
揭示氨基、酰氨基和脲基取代的3H-1,2-苯并氧杂磷杂环庚烷2-氧化物作为肿瘤相关碳酸酐酶IX和XII纳摩尔级抑制剂的潜力
期刊:ACS Medicinal Chemistry Letters
影响因子:4
doi:10.1021/acsmedchemlett.5c00099
Balašova, Anastasija; Pustenko, Aleksandrs; Angeli, Andrea; Andreucci, Elena; Biagioni, Alessio; Nocentini, Alessio; Carta, Fabrizio; Supuran, Claudiu T; Žalubovskis, Raivis