日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Potent Acridone Antimalarial against All Three Life Stages of Plasmodium

强效抗疟药吖啶酮,可对抗疟原虫所有三个生命阶段

Kancharla, Papireddy; Dodean, Rozalia A; Li, Yuexin; Zhang, Xiaowei; Kelly, Sean; Charlton, Jordan; Binauhan, Angley; Garcia, Laurize; Caridha, Diana; Madejczyk, Michael S; Jin, Xiannu; Dennis, William E; Kudyba, Karl; McEnearney, Sharon; Lee, Partricia J; Blount, Cameron; DeLuca, Jesse; Vuong, Chua; Pannone, Kristina; Dinh, Hieu T; Mdaki, Kennedy; Leed, Susan; Martin, Monica L; Pybus, Brandon S; Chimong, Anongruk; Cui, Liwang; Vega-Rodriguez, Joel; Okitwi, Martin; Kreutzfeld, Oriana; Docan, Christina; Green, Carol; Liu, Ying; Agulay, Aaron; Mirsalis, Jon; Farrell, Sarah N; McFadden, Geoffrey I; Goodman, Christopher D; Probst, Alexandra S; Nilsen, Aaron; Catteruccia, Flaminia; Rosenthal, Philip J; Riscoe, Michael; Cooper, Roland; Roth, Alison; Kelly, Jane

DDDR-05. SPATIALLY RESOLVED DRUG SENSITIVITY PROFILING IN GLIOBLASTOMA

DDDR-05. 胶质母细胞瘤的空间分辨药物敏感性分析

Kumar, Amrendra; Li, Yuexin; Dodean, Rozalia A; Roth, Alison; Caridha, Diana; Madejczyk, Michael S; Jin, Xiannu; Dennis, William E; Lee, Patricia J; Pybus, Brandon S; Martin, Monica; Pannone, Kristina; Dinh, Hieu T; Blount, Cameron; Chetree, Ravi; DeLuca, Jesse; Evans, Martin; Nadeau, Robert; Vuong, Chau; Leed, Susan; Black, Chad; Sousa, Jason; Nolan, Christina; Ceja, Frida G; Rasmussen, Stephanie A; Tumwebaze, Patrick K; Rosenthal, Philip J; Cooper, Roland A; Rottmann, Matthias; Orjuela-Sanchez, Pamela; Meister, Stephan; Winzeler, Elizabeth A; Delves, Michael J; Matthews, Holly; Baum, Jake; Kirby, Robert W; Burrows, Jeremy N; Duffy, James; Peyton, David H; Reynolds, Kevin A; Kelly, Jane X; Kancharla, Papireddy; Buck, Alicia; Lee, Sohyon; Wegmann, Rebekka; Mena, Julien; Vasella, Flavio; Friesen, Julia; Regli, Luca; Le Rhun, Emilie; Zeitlberger, Anna Maria; Neidert, Marian Christoph; Tatari, Nazanin; Hutter, Gregor; Weller, Michael; Snijder, Berend; Weiss, Tobias

Mechanisms of 8-aminoquinoline induced haemolytic toxicity in a G6PDd humanized mouse model

8-氨基喹啉在G6PDd人源化小鼠模型中诱导溶血毒性的机制

Flaherty, Siobhan; Strauch, Pamela; Maktabi, Mahdi; Pybus, Brandon S; Reichard, Gregory; Walker, Larry A; Rochford, Rosemary

Corrigendum to: Determination of Cytochrome P450 Isoenzyme 2D6 (CYP2D6) Genotypes and Pharmacogenomic Impact on Primaquine Metabolism in an Active-Duty US Military Population

更正:测定细胞色素 P450 同工酶 2D6 (CYP2D6) 基因型及其对美国现役军人伯氨喹代谢的药物基因组学影响

Spring, Michele D; Sousa, Jason C; Li, Qigui; Darko, Christian A; Morrison, Meshell N; Marcsisin, Sean R; Mills, Kristin T; Potter, Brittney M; Paolino, Kristopher M; Twomey, Patrick S; Moon, James E; Tosh, Donna M; Cicatelli, Susan B; Froude, Jeffrey W; Pybus, Brandon S; Oliver, Thomas G; Mccarthy, William F; Waters, Norman C; Smith, Philip L; Reichard, Gregory A; Bennett, Jason W

Determination of Cytochrome P450 Isoenzyme 2D6 (CYP2D6) Genotypes and Pharmacogenomic Impact on Primaquine Metabolism in an Active-Duty US Military Population

测定现役美国军人群体中细胞色素P450同工酶2D6(CYP2D6)基因型及其对伯氨喹代谢的药物基因组学影响

Spring, Michele D; Sousa, Jason C; Li, Qigui; Darko, Christian A; Morrison, Meshell N; Marcsisin, Sean R; Mills, Kristin T; Potter, Brittney M; Paolino, Kristopher M; Twomey, Patrick S; Moon, James E; Tosh, Donna M; Cicatelli, Susan B; Froude, Jeffrey W; Pybus, Brandon S; Oliver, Thomas G; McCarthy, William F; Waters, Norman C; Smith, Philip L; Reichard, Gregory A; Bennett, Jason W

Differential CYP 2D6 metabolism alters primaquine pharmacokinetics

CYP 2D6 代谢差异会改变伯氨喹的药代动力学

Potter, Brittney M J; Xie, Lisa H; Vuong, Chau; Zhang, Jing; Zhang, Ping; Duan, Dehui; Luong, Thu-Lan T; Bandara Herath, H M T; Dhammika Nanayakkara, N P; Tekwani, Babu L; Walker, Larry A; Nolan, Christina K; Sciotti, Richard J; Zottig, Victor E; Smith, Philip L; Paris, Robert M; Read, Lisa T; Li, Qigui; Pybus, Brandon S; Sousa, Jason C; Reichard, Gregory A; Marcsisin, Sean R

Differential cytochrome P450 2D metabolism alters tafenoquine pharmacokinetics

细胞色素P450 2D代谢差异改变他非诺喹的药代动力学

Vuong, Chau; Xie, Lisa H; Potter, Brittney M J; Zhang, Jing; Zhang, Ping; Duan, Dehui; Nolan, Christina K; Sciotti, Richard J; Zottig, Victor E; Nanayakkara, N P Dhammika; Tekwani, Babu L; Walker, Larry A; Smith, Philip L; Paris, Robert M; Read, Lisa T; Li, Qigui; Pybus, Brandon S; Sousa, Jason C; Reichard, Gregory A; Smith, Bryan; Marcsisin, Sean R

Tafenoquine and NPC-1161B require CYP 2D metabolism for anti-malarial activity: implications for the 8-aminoquinoline class of anti-malarial compounds

塔非诺喹和NPC-1161B需要CYP 2D代谢才能发挥抗疟活性:对8-氨基喹啉类抗疟化合物的启示

Marcsisin, Sean R; Sousa, Jason C; Reichard, Gregory A; Caridha, Diana; Zeng, Qiang; Roncal, Norma; McNulty, Ronan; Careagabarja, Julio; Sciotti, Richard J; Bennett, Jason W; Zottig, Victor E; Deye, Gregory; Li, Qigui; Read, Lisa; Hickman, Mark; Dhammika Nanayakkara, N P; Walker, Larry A; Smith, Bryan; Melendez, Victor; Pybus, Brandon S

CYP450 phenotyping and metabolite identification of quinine by accurate mass UPLC-MS analysis: a possible metabolic link to blackwater fever

利用超高效液相色谱-质谱联用技术进行CYP450表型分析和奎宁代谢物鉴定:可能与黑尿热存在代谢联系

Marcsisin, Sean R; Jin, Xiannu; Bettger, Theresa; McCulley, Nicholas; Sousa, Jason C; Shanks, G Dennis; Tekwani, Babu L; Sahu, Rajnish; Reichard, Gregory A; Sciotti, Richard J; Melendez, Victor; Pybus, Brandon S

The metabolism of primaquine to its active metabolite is dependent on CYP 2D6.

伯氨喹代谢为活性代谢物依赖于 CYP 2D6

Pybus Brandon S, Marcsisin Sean R, Jin Xiannu, Deye Gregory, Sousa Jason C, Li Qigui, Caridha Diana, Zeng Qiang, Reichard Gregory A, Ockenhouse Christian, Bennett Jason, Walker Larry A, Ohrt Colin, Melendez Victor