Identifying bias in CCR1 antagonists using radiolabelled binding, receptor internalization, β-arrestin translocation and chemotaxis assays.
利用放射性标记结合、受体内化、β-arrestin易位和趋化性试验来识别CCR1拮抗剂的偏倚
期刊:British Journal of Pharmacology
影响因子:7.7
doi:10.1111/bph.12835
Gilchrist A, Gauntner T D, Fazzini A, Alley K M, Pyen D S, Ahn J, Ha S J, Willett A, Sansom S E, Yarfi J L, Bachovchin K A, Mazzoni M R, Merritt J R