Fragment-Based Discovery of a Dual pan-RET/VEGFR2 Kinase Inhibitor Optimized for Single-Agent Polypharmacology
基于片段的发现:一种针对单一药物多药理学优化的双重泛RET/VEGFR2激酶抑制剂
期刊:Angewandte Chemie-International Edition
影响因子:16.9
doi:10.1002/anie.201501104
Frett, Brendan; Carlomagno, Francesca; Moccia, Maria Luisa; Brescia, Annalisa; Federico, Giorgia; De Falco, Valentina; Admire, Brittany; Chen, Zhongzhu; Qi, Wenqing; Santoro, Massimo; Li, Hong-yu