日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Third-generation EGFR inhibitor HS-10296 in combination with famitinib, a multi-targeted tyrosine kinase inhibitor, exerts synergistic antitumor effects through enhanced inhibition of downstream signaling in EGFR-mutant non-small cell lung cancer cells

第三代 EGFR 抑制剂 HS-10296 与多靶点酪氨酸激酶抑制剂法米替尼联合使用,可通过增强对 EGFR 突变型非小细胞肺癌细胞下游信号传导的抑制作用,发挥协同抗肿瘤作用。

Zhang, Mi; Quan, Haitian; Fu, Li; Li, Yun; Fu, Haoyu; Lou, Liguang

A modular biomimetic strategy for the synthesis of macrolide P-glycoprotein inhibitors via Rh-catalyzed C-H activation.

通过铑催化的CH活化合成大环内酯P-糖蛋白抑制剂的模块化仿生策略

Chen Lu, Quan Haitian, Xu Zhongliang, Wang Hao, Xia Yuanzhi, Lou Liguang, Yang Weibo

SHR-A1403, a novel c-mesenchymal-epithelial transition factor (c-Met) antibody-drug conjugate, overcomes AZD9291 resistance in non-small cell lung cancer cells overexpressing c-Met

SHR-A1403 是一种新型的 c-间质-上皮转化因子 (c-Met) 抗体-药物偶联物,可克服过表达 c-Met 的非小细胞肺癌细胞对 AZD9291 的耐药性。

Tong, Mengya; Gao, Mingzhao; Xu, Yongping; Fu, Li; Li, Yun; Bao, Xubin; Fu, Haoyu; Quan, Haitian; Lou, Liguang

Preclinical characterization of anlotinib, a highly potent and selective vascular endothelial growth factor receptor-2 inhibitor

安罗替尼(一种高效且选择性的血管内皮生长因子受体-2抑制剂)的临床前特性研究

Xie, Chengying; Wan, Xiaozhe; Quan, Haitian; Zheng, Mingyue; Fu, Li; Li, Yun; Lou, Liguang

STAT3 activation confers trastuzumab-emtansine (T-DM1) resistance in HER2-positive breast cancer

STAT3激活赋予HER2阳性乳腺癌对曲妥珠单抗-美坦新(T-DM1)的耐药性

Wang, Lei; Wang, Quanren; Gao, Mingzhao; Fu, Li; Li, Yun; Quan, Haitian; Lou, Liguang