日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Orthogonal IMiD-Degron Pairs Induce Selective Protein Degradation in Cells

正交IMiD-降解子对诱导细胞内选择性蛋白质降解

Brennan, Patrick J; Saunders, Rebecca E; Spanou, Mary; Singleton, Sarah E; Serafini, Marta; Sun, Liang; Heger, Guillaume P; Konopacka, Agnieszka; Beveridge, Ryan D; Taylor, C Cameron; DePaola, Peter 4th; Gordon, Laurie; Bunally, Shenaz B; Saudemont, Aurore; Benowitz, Andrew B; Martinez-Fleites, Carlos; Schmitt, Danielle L; Damoiseaux, Robert; Queisser, Markus A; An, Heeseon; Deane, Charlotte M; Hann, Michael M; Brayshaw, Lewis L; Conway, Stuart J

Optimization and Evaluation of Complementary Degrader Discovery Assays for Application in Screening.

优化和评价互补降解剂发现试验在筛选中的应用

Huchting Johanna, Weller Arjen, Schweizer Moyra, Brandt Mona, Heering Jan, Kuzikov Maria, Wolf Markus, Reinshagen Jeanette, Queisser Markus A, Gribbon Philip, Zaliani Andrea, Pless Ole, Kannt Aimo

Corrigendum: miR-182 integrates apoptosis, growth, and differentiation programs in glioblastoma

更正:miR-182整合胶质母细胞瘤中的细胞凋亡、生长和分化程序

Kouri, Fotini M; Hurley, Lisa A; Daniel, Weston L; Day, Emily S; Hua, Youjia; Hao, Liangliang; Peng, Chian-Yu; Merkel, Timothy J; Queisser, Markus A; Ritner, Carissa; Zhang, Hailei; James, C David; Sznajder, Jacob I; Chin, Lynda; Giljohann, David A; Kessler, John A; Peter, Marcus E; Mirkin, Chad A; Stegh, Alexander H

Antibody-Proteolysis Targeting Chimera Conjugate Enables Selective Degradation of Receptor-Interacting Serine/Threonine-Protein Kinase 2 in HER2+ Cell Lines

抗体-蛋白水解靶向嵌合偶联物可选择性降解HER2+细胞系中的受体相互作用丝氨酸/苏氨酸蛋白激酶2

Chan, Karina; Sathyamurthi, Preethi Soundarya; Queisser, Markus A; Mullin, Michael; Shrives, Harry; Coe, Diane M; Burley, Glenn A

HIF and HOIL-1L-mediated PKCζ degradation stabilizes plasma membrane Na,K-ATPase to protect against hypoxia-induced lung injury

HIF 和 HOIL-1L 介导的 PKCζ 降解可稳定质膜 Na,K-ATPase,从而保护肺免受缺氧引起的损伤。

Magnani, Natalia D; Dada, Laura A; Queisser, Markus A; Brazee, Patricia L; Welch, Lynn C; Anekalla, Kishore R; Zhou, Guofei; Vagin, Olga; Misharin, Alexander V; Budinger, G R Scott; Iwai, Kazuhiro; Ciechanover, Aaron J; Sznajder, Jacob I

HOIL-1L functions as the PKCζ ubiquitin ligase to promote lung tumor growth

HOIL-1L 作为 PKCζ 泛素连接酶,促进肺肿瘤生长

Queisser, Markus A; Dada, Laura A; Deiss-Yehiely, Nimrod; Angulo, Martin; Zhou, Guofei; Kouri, Fotini M; Knab, Lawrence M; Liu, Jing; Stegh, Alexander H; DeCamp, Malcolm M; Budinger, G R Scott; Chandel, Navdeep S; Ciechanover, Aaron; Iwai, Kazuhiro; Sznajder, Jacob I