日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

An allosteric inhibitor of the Zika virus NS2B-NS3 protease with oral efficacy in mouse models

一种寨卡病毒NS2B-NS3蛋白酶的变构抑制剂,在小鼠模型中具有口服疗效。

Ontoria, Jesus M; Torrente, Esther; Missineo, Antonino; Alli, Cristina; Graziani, Rita; Conti, Silvia; Bisbocci, Monica; Quotadamo, Antonio; Ferrigno, Federica; Corio, Alessandra; Ievoli, Giovanni; Bencheva, Leda; Amaudrut, Jérôme; Vasile, Silvana; Beghetto, Elisa; Paolini, Chantal; Alaimo, Nadine; Veneziano, Maria; Nibbio, Martina; Orsale, Maria V; Proto, Giulia; Colaceci, Fabrizio; Orsatti, Laura; Pucci, Vincenzo; Di Fabio, Romano; Tomei, Licia; Montalbetti, Christian; Bresciani, Alberto; Toniatti, Carlo; Paonessa, Giacomo

High-Throughput Phenotypic Screening and Machine Learning Methods Enabled the Selection of Broad-Spectrum Low-Toxicity Antitrypanosomatidic Agents

高通量表型筛选和机器学习方法能够选择广谱低毒抗锥虫病药物

Pasquale Linciano, Antonio Quotadamo, Rosaria Luciani, Matteo Santucci, Kimberley M Zorn, Daniel H Foil, Thomas R Lane, Anabela Cordeiro da Silva, Nuno Santarem, Carolina B Moraes, Lucio Freitas-Junior, Ulrike Wittig, Wolfgang Mueller, Michele Tonelli, Stefania Ferrari, Alberto Venturelli, Sheraz Gu

Identification of novel anti-amoebic pharmacophores from kinase inhibitor chemotypes

从激酶抑制剂化学类型中鉴定新型抗阿米巴药效团

Ferrins, Lori; Buskes, Melissa J; Kapteyn, Madison M; Engels, Hannah N; Enos, Suzanne E; Lu, Chenyang; Klug, Dana M; Singh, Baljinder; Quotadamo, Antonio; Bachovchin, Kelly; Tear, Westley F; Spaulding, Andrew E; Forbes, Katherine C; Bag, Seema; Rivers, Mitch; LeBlanc, Catherine; Burchfield, Erin; Armand, Jeremy R; Diaz-Gonzalez, Rosario; Ceballos-Perez, Gloria; García-Hernández, Raquel; Pérez-Moreno, Guiomar; Bosch-Navarrete, Cristina; Ruiz-Pérez, Luis Miguel; Gamarro, Francisco; González-Pacanowska, Dolores; Navarro, Miguel; Mensa-Wilmot, Kojo; Pollastri, Michael P; Kyle, Dennis E; Rice, Christopher A

Corrigendum: Identification of novel anti-amoebic pharmacophores from kinase inhibitor chemotypes

更正:从激酶抑制剂化学类型中鉴定新型抗阿米巴药效团

Ferrins, Lori; Buskes, Melissa J; Kapteyn, Madison M; Engels, Hannah N; Enos, Suzanne E; Lu, Chenyang; Klug, Dana M; Singh, Baljinder; Quotadamo, Antonio; Bachovchin, Kelly; Tear, Westley F; Spaulding, Andrew E; Forbes, Katherine C; Bag, Seema; Rivers, Mitch; LeBlanc, Catherine; Burchfield, Erin; Armand, Jeremy R; Diaz-Gonzalez, Rosario; Ceballos-Perez, Gloria; García-Hernández, Raquel; Pérez-Moreno, Guiomar; Bosch-Navarrete, Cristina; Gómez-Liñán, Claudia; Ruiz-Pérez, Luis Miguel; Gamarro, Francisco; González-Pacanowska, Dolores; Navarro, Miguel; Mensa-Wilmot, Kojo; Pollastri, Michael P; Kyle, Dennis E; Rice, Christopher A

Structure-Property Optimization of a Series of Imidazopyridines for Visceral Leishmaniasis

一系列咪唑并吡啶类化合物的结构-性质优化及其在内脏利什曼病中的应用

Dichiara, Maria; Simpson, Quillon J; Quotadamo, Antonio; Jalani, Hitesh B; Huang, Anson X; Millard, Caroline C; Klug, Dana M; Tse, Edwin G; Todd, Matthew H; Silva, Daniel Gedder; da Silva Emery, Flavio; Carlson, J Eric; Zheng, Shao-Liang; Vleminckx, Margot; Matheeussen, An; Caljon, Guy; Pollastri, Michael P; Sjö, Peter; Perry, Benjamin; Ferrins, Lori

Multitarget, Selective Compound Design Yields Potent Inhibitors of a Kinetoplastid Pteridine Reductase 1

多靶点选择性化合物设计获得了强效的动质体蝶呤还原酶抑制剂 1

Pöhner, Ina; Quotadamo, Antonio; Panecka-Hofman, Joanna; Luciani, Rosaria; Santucci, Matteo; Linciano, Pasquale; Landi, Giacomo; Di Pisa, Flavio; Dello Iacono, Lucia; Pozzi, Cecilia; Mangani, Stefano; Gul, Sheraz; Witt, Gesa; Ellinger, Bernhard; Kuzikov, Maria; Santarem, Nuno; Cordeiro-da-Silva, Anabela; Costi, Maria P; Venturelli, Alberto; Wade, Rebecca C

Destabilizers of the thymidylate synthase homodimer accelerate its proteasomal degradation and inhibit cancer growth

胸苷酸合酶同型二聚体的不稳定剂会加速其蛋白酶体降解并抑制癌症生长

Luca Costantino, Stefania Ferrari, Matteo Santucci, Outi M H Salo-Ahen, Emanuele Carosati, Silvia Franchini, Angela Lauriola, Cecilia Pozzi, Matteo Trande, Gaia Gozzi, Puneet Saxena, Giuseppe Cannazza, Lorena Losi, Daniela Cardinale, Alberto Venturelli, Antonio Quotadamo, Pasquale Linciano, Lorenzo

New Insights into Bioactive Compounds from the Medicinal Plant Spathodea campanulata P. Beauv. and Their Activity against Helicobacter pylori

对药用植物 Spathodea campanulata P. Beauv. 的生物活性化合物及其抗幽门螺杆菌活性的新见解

Corinne Raïssa Ngnameko, Lucia Marchetti, Barbara Zambelli, Antonio Quotadamo, Davide Roncarati, Davide Bertelli, Frederic Nico Njayou, Stella I Smith, Paul F Moundipa, Maria Paola Costi, Federica Pellati