日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Preclinical characterization of an intravenous coronavirus 3CL protease inhibitor for the potential treatment of COVID19

对一种用于治疗 COVID-19 的静脉注射冠状病毒 3CL 蛋白酶抑制剂进行临床前表征

Britton Boras # ,Rhys M Jones # ,Brandon J Anson ,Dan Arenson ,Lisa Aschenbrenner ,Malina A Bakowski ,Nathan Beutler ,Joseph Binder ,Emily Chen ,Heather Eng ,Holly Hammond ,Jennifer Hammond ,Robert E Haupt ,Robert Hoffman ,Eugene P Kadar ,Rob Kania ,Emi Kimoto ,Melanie G Kirkpatrick ,Lorraine Lanyon ,Emma K Lendy ,Jonathan R Lillis ,James Logue ,Suman A Luthra ,Chunlong Ma ,Stephen W Mason ,Marisa E McGrath ,Stephen Noell ,R Scott Obach ,Matthew N O' Brien ,Rebecca O'Connor ,Kevin Ogilvie ,Dafydd Owen ,Martin Pettersson ,Matthew R Reese ,Thomas F Rogers ,Romel Rosales ,Michelle I Rossulek ,Jean G Sathish ,Norimitsu Shirai ,Claire Steppan ,Martyn Ticehurst ,Lawrence W Updyke ,Stuart Weston ,Yuao Zhu ,Kris M White ,Adolfo García-Sastre ,Jun Wang ,Arnab K Chatterjee ,Andrew D Mesecar ,Matthew B Frieman ,Annaliesa S Anderson ,Charlotte Allerton

Development of Robust Quantitative Structure-Activity Relationship Models for CYP2C9, CYP2D6, and CYP3A4 Catalysis and Inhibition

开发针对 CYP2C9、CYP2D6 和 CYP3A4 催化和抑制的稳健定量结构-活性关系模型

Eric Gonzalez, Sankalp Jain, Pranav Shah, Nao Torimoto-Katori, Alexey Zakharov, Ðắc-Trung Nguyễn, Srilatha Sakamuru, Ruili Huang, Menghang Xia, R Scott Obach, Cornelis E C A Hop, Anton Simeonov, Xin Xu

An Automated High-Throughput Metabolic Stability Assay Using an Integrated High-Resolution Accurate Mass Method and Automated Data Analysis Software

使用集成高分辨率精确质量法和自动数据分析软件进行自动化高通量代谢稳定性分析

Pranav Shah, Edward Kerns, Dac-Trung Nguyen, R Scott Obach, Amy Q Wang, Alexey Zakharov, John McKew, Anton Simeonov, Cornelis E C A Hop, Xin Xu

2-aryloxy-4-alkylaminopyridines: discovery of novel corticotropin-releasing factor 1 antagonists

2-芳氧基-4-烷基氨基吡啶:发现新型促皮质素释放因子 1 拮抗剂

Yuhpyng L Chen, R Scott Obach, John Braselton, Michael L Corman, James Forman, Jody Freeman, Randall J Gallaschun, Robert Mansbach, Anne W Schmidt, Jeffrey S Sprouse, F David Tingley Iii, Elizabeth Winston, David W Schulz