NVL-655 Is a Selective and Brain-Penetrant Inhibitor of Diverse ALK-Mutant Oncoproteins, Including Lorlatinib-Resistant Compound Mutations
NVL-655 是一种选择性、脑渗透性抑制剂,可抑制多种 ALK 突变癌蛋白,包括劳拉替尼耐药化合物突变
期刊:Cancer Discovery
影响因子:29.7
doi:10.1158/2159-8290.CD-24-0231
Jessica J Lin #, Joshua C Horan #, Anupong Tangpeerachaikul #, Aurélie Swalduz, Augusto Valdivia, Melissa L Johnson, Benjamin Besse, D Ross Camidge, Toshio Fujino, Satoshi Yoda, Linh Nguyen-Phuong, Hayato Mizuta, Ludovic Bigot, Catline Nobre, Jii Bum Lee, Mi Ra Yu, Scot Mente, Yuting Sun, Nancy E Ko