日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Clinical and Physiologically Based Pharmacokinetic Model Evaluations of Adagrasib Drug-Drug Interactions

基于临床和生理的药代动力学模型对阿达格拉西布药物相互作用的评价

Cilliers, Cornelius; Howgate, Eleanor; Jones, Hannah M; Rahbaek, Lisa; Tran, Jonathan Q

Discovery of Pyridopyrimidinones that Selectively Inhibit the H1047R PI3Kα Mutant Protein

发现能选择性抑制H1047R PI3Kα突变蛋白的吡啶并嘧啶酮类化合物

Ketcham, John M; Harwood, Stephen J; Aranda, Ruth; Aloiau, Athenea N; Bobek, Briana M; Briere, David M; Burns, Aaron C; Caddell Haatveit, Kersti; Calinisan, Andrew; Clarine, Jeffery; Elliott, Adam; Engstrom, Lars D; Gunn, Robin J; Ivetac, Anthony; Jones, Benjamin; Kuehler, Jon; Lawson, J David; Nguyen, Natalie; Parker, Cody; Pearson, Kelly E; Rahbaek, Lisa; Saechao, Barbara; Wang, Xiaolun; Waters, Anna; Waters, Laura; Watkins, Ashlee H; Olson, Peter; Smith, Christopher R; Christensen, James G; Marx, Matthew A

The SOS1 Inhibitor MRTX0902 Blocks KRAS Activation and Demonstrates Antitumor Activity in Cancers Dependent on KRAS Nucleotide Loading

SOS1 抑制剂 MRTX0902 可阻断 KRAS 激活,并在依赖 KRAS 核苷酸加载的癌症中表现出抗肿瘤活性

Niranjan Sudhakar, Larry Yan, Fadia Qiryaqos, Lars D Engstrom, Jade Laguer, Andrew Calinisan, Allan Hebbert, Laura Waters, Krystal Moya, Vickie Bowcut, Laura Vegar, John M Ketcham, Anthony Ivetac, Christopher R Smith, J David Lawson, Lisa Rahbaek, Jeffrey Clarine, Natalie Nguyen, Barbara Saechao, Co

Design and Immunological Validation of Macaca fascicularis Papillomavirus Type 3 Based Vaccine Candidates in Outbred Mice: Basis for Future Testing of a Therapeutic Papillomavirus Vaccine in NHPs

食蟹猴乳头瘤病毒 3 型疫苗候选物的设计和在杂交小鼠中的免疫学验证:为未来在 NHP 中测试治疗性乳头瘤病毒疫苗奠定基础

Patrick Neckermann, Ditte Rahbaek Boilesen, Torsten Willert, Cordula Pertl, Silke Schrödel, Christian Thirion, Benedikt Asbach, Peter Johannes Holst, Ralf Wagner