日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

A µ-opioid receptor superagonist analgesic with minimal adverse effects

一种μ-阿片受体超激动剂镇痛药,不良反应极小

Gomez, Juan L; Ventriglia, Emilya N; Frangos, Zachary J; Sulima, Agnieszka; Robertson, Michael J; Sacco, Michael D; Budinich, Reece C; Giosan, Ilinca M; Xie, Tongzhen; Solis, Oscar; Tischer, Anna E; Bossert, Jennifer M; Caldwell, Kiera E; Bonbrest, Hannah; Essmann, Amelie; Garçon-Poca, Zelai M; Choi, Shinbe; Noya, Michael R; Limiac, Feonil; Arce, Ali; Glatfelter, Grant C; Robinson, Margaret; Chen, Li; Mullarkey, Angelina A; Brademan, Dain R; Enten, Garrett; Dunne, William; Quiroz, César; Schoenborn, Ingrid; Lee, Chae Bin; Rais, Rana; Holt, Daniel P; Dannals, Robert F; Shi, Lei; Hüttenhain, Ruth; Ferré, Sergi; Kiyatkin, Eugene; Bonaventura, Jordi; Shaham, Yavin; Zachariou, Venetia; Baumann, Michael H; Skiniotis, Georgios; Rice, Kenner C; Michaelides, Michael

Tailoring cariprazine for dual disorders via secondary pharmacophore optimization

通过二级药效团优化来定制卡利拉嗪用于治疗双重疾病

Vogt, Caleb D; Sanchez, Julie; Bonifazi, Alessandro; Saab, Elizabeth; Ranjit, Arina; Rais, Rana; Lane, J Robert; Newman, Amy Hauck

Dendrimer-Conjugated Glutamine Antagonist, D-TTM020, Ameliorates Brain Immune Dysregulation and Improves Neurobehavioral Deficits in the Mecp2-Deficient Mouse Model

树状聚合物偶联的谷氨酰胺拮抗剂D-TTM020可改善Mecp2缺陷小鼠模型的脑免疫失调并改善其神经行为缺陷。

Vyas, Preeti; Khoury, Elizabeth Smith; Sah, Nirnath; Sharma, Anjali; Allende Labastida, Javier; Wilkinson, Elizabeth L; Lac, Kathleen; Damiba, Nerketa N L; Fowler, Amanda; Liu, Jinhuan; Bedner, Ashley; Majer, Pavel; Tichý, Tomás; Thomas, Ajit G; Rais, Rana; Slusher, Barbara S; Kannan, Rangaramanujam M; Kannan, Sujatha

Microglial-Targeted GCPII Inhibition Reverses Neurocognitive Impairment and Synaptic Loss After EcoHIV Infection.

靶向小胶质细胞的 GCPII 抑制可逆转 EcoHIV 感染后的神经认知障碍和突触丢失。

Zheng Yuxin, Huang Meixiang, Maragakis R Michael, Pietri Peter, Su Yu, Alt Jesse, Tenora Lukáš, Liyanage Wathsala, Wu Ying, Thomas Mary-Anne, Kannan Rangaramanujam M, Zhu Xiaolei, Rais Rana, Slusher Barbara S

A Star-PEGylation Strategy to Improve Testosterone Pharmacokinetics

星形聚乙二醇化策略改善睾酮药代动力学

Lee, Chae Bin; Tenora, Lukáš; Zhang, Ruoning; Ranjit, Arina; Markowski, Mark C; Slusher, Barbara S; Rais, Rana

Discovery of N-Acetyltransferase 8-Like (NAT8L) inhibitors based on a N-Acylated (Piperidin-3-ylmethyl)-1,2,4-Oxadiazole Scaffold

基于 N-酰化(哌啶-3-基甲基)-1,2,4-恶二唑骨架的 N-乙酰转移酶 8 样(NAT8L)抑制剂的发现

Nayeen, Md Junayed; Thomas, Ajit G; Kundu, Biswajit; Carlyle, Evan; Hin, Niyada; Hin, Philana; Pal, Arindom; Paule, James; Rais, Rana; Slusher, Barbara S; Tsukamoto, Takashi

Bioisosteric Replacement of Amides with 1,2,3-Triazoles Improves Dopamine D4 Receptor Ligand Pharmacokinetics

用1,2,3-三唑类化合物生物等排取代酰胺类化合物可改善多巴胺D4受体配体的药代动力学

Alkhatib, Mohammad; Jakobs, Franziska M; Hanson, John N; Nilson, Ashley N; Moritz, Amy E; Li, Tian; Faibille, Afua B; Bourn, Lindsay A; Ramdhan, Peter A; Ricchezza, Joseph 4th; Jordan, Shannon; Panasis, Diandra; Nguyen, Norman; Kasarla, Nitish; Wang, Bryant; Garcia, Sergio Sola; Saez, Julianna; Paule, James; Lee, Chae Bin; Rais, Rana; Slusher, Barbara S; Sibley, David R; Li, Chenglong; Keck, Thomas M; Boateng, Comfort A

Targeting NAAG metabolism restores cognition and synaptic integrity in EcoHIV-infected mice

靶向NAAG代谢可恢复EcoHIV感染小鼠的认知功能和突触完整性。

Zheng, Yuxin; Huang, Meixiang; Maragakis, R Michael; Pietri, Peter; Su, Yu; Alt, Jesse; Wu, Ying; Finney, Colin; Peters, Diane E; Zhu, Xiaolei; Rais, Rana; Slusher, Barbara S

Translin deletion impairs cocaine-induced locomotor sensitization and RGS8 expression in the nucleus accumbens

Translin基因缺失会损害伏隔核中可卡因诱导的运动敏化和RGS8表达。

Fu, Xiu-Ping; Wu, Ren-Kun; Shah, Aparna P; Ladenheim, Bruce; Alt, Jesse; Cadet, Jean Lud; Rais, Rana; Chandra, Ramesh; Cen, Xiao-Bo; Baraban, Jay M

JHU-2545 preferentially shields salivary glands and kidneys during PSMA-targeted imaging

在PSMA靶向成像过程中,JHU-2545优先保护唾液腺和肾脏。

Nedelcovych, Michael T; Dash, Ranjeet P; Wu, Ying; Choi, Eun Yong; Lapidus, Rena S; Majer, Pavel; Jančařík, Andrej; Abou, Diane; Penet, Marie-France; Nikolopoulou, Anastasia; Amor-Coarasa, Alex; Babich, John; Thorek, Daniel L; Rais, Rana; Kratochwil, Clemens; Slusher, Barbara S