Chirality matters: stereo-defined phosphorothioate linkages at the termini of small interfering RNAs improve pharmacology in vivo
手性很重要:小干扰 RNA 末端的立体定义的硫代磷酸酯键可改善体内药理学
期刊:Nucleic Acids Research
影响因子:16.6
doi:10.1093/nar/gkab544
Hartmut Jahns, Nate Taneja, Jennifer L S Willoughby, Masaaki Akabane-Nakata, Christopher R Brown, Tuyen Nguyen, Anna Bisbe, Shigeo Matsuda, Matt Hettinger, Rajar M Manoharan, Kallanthottathil G Rajeev, Martin A Maier, Ivan Zlatev, Klaus Charisse, Martin Egli, Muthiah Manoharan