日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Structure-Guided Design of ISOX-DUAL-Based Degraders Targeting BRD4 and CBP/EP300: A Case of Degrader Collapse.

基于 ISOX-DUAL 的结构导向降解剂设计:针对 BRD4 和 CBP/EP300 的降解剂崩溃案例

Edmonds Anthony K, Balourdas Dimitrios-Ilias, Marsh Graham P, Felix Robert, Brasher Bradley, Cooper Jeff, Graber-Feesl Cari, Kollareddy Madhu, Malik Karim, Stewart Helen, Chevassut Timothy J T, Lineham Ella, Morley Simon, Fedorov Oleg, Bennett James, Rajasekaran Mohan B, Ojeda Samuel, Harrison Drew A, Ott Christopher J, Joerger Andreas C, Maple Hannah J, Spencer John

Crystal structure and metal binding properties of the periplasmic iron component EfeM from Pseudomonas syringae EfeUOB/M iron-transport system

丁香假单胞菌EfeUOB/M铁转运系统周质铁组分EfeM的晶体结构和金属结合特性

Rajasekaran, Mohan B; Hussain, Rohanah; Siligardi, Giuliano; Andrews, Simon C; Watson, Kimberly A

A first generation inhibitor of human Greatwall kinase, enabled by structural and functional characterisation of a minimal kinase domain construct

通过对最小激酶结构域构建体进行结构和功能表征,开发出第一代人长城激酶抑制剂。

Ocasio, Cory A; Rajasekaran, Mohan B; Walker, Sarah; Le Grand, Darren; Spencer, John; Pearl, Frances M G; Ward, Simon E; Savic, Velibor; Pearl, Laurence H; Hochegger, Helfrid; Oliver, Antony W