日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Accelerating Generic Long-Acting Antiretrovirals for Global HIV Treatment: Workshop Findings and a Roadmap to Access

加速推广通用长效抗逆转录病毒药物以用于全球艾滋病治疗:研讨会成果及获取路线图

Arshad, Usman; Gaayeb, Lobna; Pertinez, Henry; Rajoli, Rajith K R; Watkins, Melynda; Nimbolkar, Parag; Perazzolo, Simone; Pagi, Bharat; Wensing, Annemarie; Khoo, Saye; Boffito, Marta; Holm, René; Panos, Zack; Mahaka, Imelda; Venter, Francois; Kottiri, Benny; Crawford, Keith W; Ho, Rodney J Y; Clayden, Polly; Domanico, Paul; Struble, Kimberly; Owen, Andrew; Flexner, Charles

Lack of antiviral activity of probenecid in vitro and in Syrian golden hamsters

丙磺舒在体外和叙利亚金黄仓鼠中缺乏抗病毒活性

Helen J Box, Joanne Sharp, Shaun H Pennington, Edyta Kijak, Lee Tatham, Claire H Caygill, Rose C Lopeman, Laura N Jeffreys, Joanne Herriott, Megan Neary, Anthony Valentijn, Henry Pertinez, Paul Curley, Usman Arshad, Rajith K R Rajoli, Dirk Jochmans, Laura Vangeel, Johan Neyts, Eric Chatelain, Fanny

Assessment of Favipiravir and Remdesivir in Combination for SARS-CoV-2 Infection in Syrian Golden Hamsters

评估法匹拉韦和瑞德西韦联合治疗叙利亚金仓鼠SARS-CoV-2感染的疗效

Neary, Megan; Gallardo-Toledo, Eduardo; Sharp, Joanne; Herriott, Joanne; Kijak, Edyta; Bramwell, Chloe; Cox, Helen; Tatham, Lee; Box, Helen; Curley, Paul; Arshad, Usman; Rajoli, Rajith K R; Pertinez, Henry; Valentijn, Anthony; Pennington, Shaun H; Caygill, Claire H; Lopeman, Rose C; Biagini, Giancarlo A; Kipar, Anja; Stewart, James P; Owen, Andrew

Physiologically Based Pharmacokinetic Modelling of Cabotegravir Microarray Patches in Rats and Humans

基于生理的卡博特韦微阵列贴剂在大鼠和人体内的药代动力学模型

Kinvig, Hannah; Rajoli, Rajith K R; Pertinez, Henry; Vora, Lalitkumar K; Volpe-Zanutto, Fabiana; Donnelly, Ryan F; Rannard, Steve; Flexner, Charles; Siccardi, Marco; Owen, Andrew

Evaluation of Nafamostat as Chemoprophylaxis for SARS-CoV-2 Infection in Hamsters

评估萘莫司他作为SARS-CoV-2感染化学预防药物在仓鼠中的应用

Neary, Megan; Sharp, Joanne; Gallardo-Toledo, Eduardo; Herriott, Joanne; Kijak, Edyta; Bramwell, Chloe; Cox, Helen; Tatham, Lee; Box, Helen; Curley, Paul; Arshad, Usman; Rajoli, Rajith K R; Pertinez, Henry; Valentijn, Anthony; Dhaliwal, Kevin; Mc Caughan, Frank; Hobson, James; Rannard, Steve; Kipar, Anja; Stewart, James P; Owen, Andrew

Chemoprophylactic Assessment of Combined Intranasal SARS-CoV-2 Polymerase and Exonuclease Inhibition in Syrian Golden Hamsters

叙利亚金仓鼠鼻内联合应用SARS-CoV-2聚合酶和核酸外切酶抑制剂的化学预防效果评估

Gallardo-Toledo, Eduardo; Neary, Megan; Sharp, Joanne; Herriott, Joanne; Kijak, Edyta; Bramwell, Chloe; Curley, Paul; Arshad, Usman; Pertinez, Henry; Rajoli, Rajith K R; Valentijn, Anthony; Cox, Helen; Tatham, Lee; Kipar, Anja; Stewart, James P; Owen, Andrew

Unlike Chloroquine, Mefloquine Inhibits SARS-CoV-2 Infection in Physiologically Relevant Cells

与氯喹不同,甲氟喹能抑制生理相关细胞中的SARS-CoV-2感染。

Sacramento, Carolina Q; Fintelman-Rodrigues, Natalia; Dias, Suelen S G; Temerozo, Jairo R; Da Silva, Aline de Paula D; da Silva, Carine S; Blanco, Camilla; Ferreira, André C; Mattos, Mayara; Soares, Vinicius C; Pereira-Dutra, Filipe; Miranda, Milene Dias; Barreto-Vieira, Debora F; da Silva, Marcos Alexandre N; Santos, Suzana S; Torres, Mateo; Chaves, Otávio Augusto; Rajoli, Rajith K R; Paccanaro, Alberto; Owen, Andrew; Bou-Habib, Dumith Chequer; Bozza, Patrícia T; Souza, Thiago Moreno L

Physiologically based pharmacokinetic modeling for dose optimization of quinine-phenobarbital coadministration in patients with cerebral malaria

基于生理的药代动力学模型用于优化奎宁-苯巴比妥联合用药治疗脑型疟疾患者的剂量

Sae-Heng, Teerachat; Rajoli, Rajith Kumar Reddy; Siccardi, Marco; Karbwang, Juntra; Na-Bangchang, Kesara

Lack of antiviral activity of probenecid in Vero E6 cells and Syrian golden hamsters: a need for better understanding of inter-lab differences in preclinical assays

丙磺舒在 Vero E6 细胞和叙利亚金黄仓鼠中缺乏抗病毒活性:需要更好地了解临床前检测中实验室间的差异

Helen Box, Shaun H Pennington, Edyta Kijak, Lee Tatham, Claire H Caygill, Rose C Lopeman, Laura N Jeffreys, Joanne Herriott, Joanne Sharp, Megan Neary, Anthony Valentijn, Henry Pertinez, Paul Curley, Usman Arshad, Rajith Kr Rajoli, Steve Rannard, James P Stewart, Giancarlo A Biagini, Andrew Owen

In vitro antiviral activity of the anti-HCV drugs daclatasvir and sofosbuvir against SARS-CoV-2, the aetiological agent of COVID-19

体外抗HCV药物达克拉他韦和索非布韦对SARS-CoV-2(COVID-19的病原体)的抗病毒活性

Sacramento, Carolina Q; Fintelman-Rodrigues, Natalia; Temerozo, Jairo R; Da Silva, Aline de Paula Dias; Dias, Suelen da Silva Gomes; da Silva, Carine Dos Santos; Ferreira, André C; Mattos, Mayara; Pão, Camila R R; de Freitas, Caroline S; Soares, Vinicius Cardoso; Hoelz, Lucas Villas Bôas; Fernandes, Tácio Vinício Amorim; Branco, Frederico Silva Castelo; Bastos, Mônica Macedo; Boechat, Núbia; Saraiva, Felipe B; Ferreira, Marcelo Alves; Jockusch, Steffen; Wang, Xuanting; Tao, Chuanjuan; Chien, Minchen; Xie, Wei; Patel, Dinshaw; Garzia, Aitor; Tuschl, Thomas; Russo, James J; Rajoli, Rajith K R; Pedrosa, Carolina S G; Vitória, Gabriela; Souza, Letícia R Q; Goto-Silva, Livia; Guimarães, Marilia Zaluar; Rehen, Stevens K; Owen, Andrew; Bozza, Fernando A; Bou-Habib, Dumith Chequer; Ju, Jingyue; Bozza, Patrícia T; Souza, Thiago Moreno L