日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

ADT-030, a novel PDE10 inhibitor, demonstrates potent antitumor activity in pancreatic ductal adenocarcinoma

ADT-030 是一种新型 PDE10 抑制剂,在胰腺导管腺癌中表现出强大的抗肿瘤活性。

Bandi, Dhana Sekhar Reddy; Nagaraju, Ganji Purnachandra; Sarvesh, Sujith; Foote, Jeremy B; Keeton, Adam B; Chen, Xi; Ramirez-Alcantara, Veronica; Holmes, Thomas; Akce, Mehmet; Singh, Anju; Powell, Craig M; Behera, Santosh; Azmi, Asfar S; Nurmemmedov, Elmar; Babic, Ivan; Gorman, Gregory S; Coward, Lori; Buchsbaum, Donald J; Maxuitenko, Yulia Y; Piazza, Gary A; El-Rayes, Bassel F

A Pan-RAS Inhibitor with a Unique Mechanism of Action Blocks Tumor Growth and Induces Antitumor Immunity in Gastrointestinal Cancer.

一种具有独特作用机制的泛 RAS 抑制剂可抑制肿瘤生长并诱导胃肠道癌症的抗肿瘤免疫

Foote Jeremy B, Mattox Tyler E, Keeton Adam B, Chen Xi, Smith Forrest T, Berry Kristy, Holmes Thomas W, Wang Junwei, Huang Chung-Hui, Ward Antonio, Mitra Amit K, Ramirez-Alcantara Veronica, Hardy Cherlene, Fleten Karianne G, Flatmark Kjersti, Yoon Karina J, Sarvesh Sujith, Nagaraju Ganji P, Bandi Dhana Sekhar Reddy, Maxuitenko Yulia Y, Valiyaveettil Jacob, Carstens Julienne L, Buchsbaum Donald J, Yang Jennifer, Zhou Gang, Nurmemmedov Elmar, Babic Ivan, Gaponeko Vadim, Abdelkarim Hazem, Boyd Michael R, Gorman Greg, Manne Upender, Bae Sejong, El-Rayes Bassel F, Piazza Gary A

A Novel Pan-RAS Inhibitor with a Unique Mechanism of Action Blocks Tumor Growth in Mouse Models of GI Cancer

一种具有独特作用机制的新型泛RAS抑制剂可抑制小鼠胃肠道癌症模型中的肿瘤生长

Foote, Jeremy B; Mattox, Tyler E; Keeton, Adam B; Chen, Xi; Smith, Forrest; Berry, Kristy L; Holmes, Thomas; Wang, Junwei; Huang, Chung-Hui; Ward, Antonio B; Mitra, Amit K; Ramirez-Alcantara, Veronica; Hardy, Cherlene; Fleten, Karrianne G; Flatmark, Kjersti; Yoon, Karina J; Sarvesh, Sujith; Nagaraju, Ganji Purnachandra; Bandi, Dhana Sekhar Reddy; Maxuitenko, Yulia Y; Valiyaveettil, Jacob; Carstens, Julienne L; Buchsbaum, Donald J; Yang, Jennifer; Zhou, Gang; Nurmemmedov, Elmar; Babic, Ivan; Gaponenko, Vadim; Abdelkarim, Hazem; Boyd, Michael R; Gorman, Gregory S; Manne, Upender; Bae, Sejong; El-Rayes, Bassel F; Piazza, Gary A