AKT Degradation Selectively Inhibits the Growth of PI3K/PTEN Pathway-Mutant Cancers with Wild-Type KRAS and BRAF by Destabilizing Aurora Kinase B
AKT降解通过使Aurora激酶B不稳定,选择性地抑制具有野生型KRAS和BRAF的PI3K/PTEN通路突变型癌症的生长。
期刊:Cancer Discovery
影响因子:29.7
doi:10.1158/2159-8290.CD-20-0815
Jia Xu # ,Xufen Yu # ,Tiphaine C Martin ,Ankita Bansal ,Kakit Cheung ,Abigail Lubin ,Elias Stratikopoulos ,Kaitlyn M Cahuzac ,Li Wang ,Ling Xie ,Royce Zhou ,Yudao Shen ,Xuewei Wu ,Shen Yao ,Ruifang Qiao ,Poulikos I Poulikakos ,Xian Chen ,Jing Liu ,Jian Jin ,Ramon Parsons