日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Correction: Progress in the discovery and development of anticancer agents from marine cyanobacteria

更正:海洋蓝藻抗癌药物的发现和开发进展

Luesch, Hendrik; Ellis, Emma K; Chen, Qi-Yin; Ratnayake, Ranjala

Progress in the discovery and development of anticancer agents from marine cyanobacteria

海洋蓝藻抗癌药物的发现与开发进展

Luesch, Hendrik; Ellis, Emma K; Chen, Qi-Yin; Ratnayake, Ranjala

Morphological profiling for drug discovery in the era of deep learning

深度学习时代药物发现的形态学分析

Tang, Qiaosi; Ratnayake, Ranjala; Seabra, Gustavo; Jiang, Zhe; Fang, Ruogu; Cui, Lina; Ding, Yousong; Kahveci, Tamer; Bian, Jiang; Li, Chenglong; Luesch, Hendrik; Li, Yanjun

Biosynthesis of Dolastatin 10 in Marine Cyanobacteria, a Prototype for Multiple Approved Cancer Drugs

海洋蓝藻中多拉司他汀10的生物合成,是多种已获批准的抗癌药物的原型

Kallifidas, Dimitris; Dhakal, Dipesh; Chen, Manyun; Chen, Qi-Yin; Kokkaliari, Sofia; Colon Rosa, Nicole A; Ratnayake, Ranjala; Bruner, Steven D; Paul, Valerie J; Ding, Yousong; Luesch, Hendrik

Epigenetic small-molecule screen for inhibition and reversal of acinar ductal metaplasia in mouse pancreatic organoids

表观遗传小分子筛选抑制和逆转小鼠胰腺类器官中的腺泡导管化生

Kalina R Atanasova #, Corey M Perkins #, Ranjala Ratnayake, Jinmai Jiang, Qi-Yin Chen, Thomas D Schmittgen, Hendrik Luesch

Chemical Genetics in C. elegans Identifies Anticancer Mycotoxins Chaetocin and Chetomin as Potent Inducers of a Nuclear Metal Homeostasis Response.

秀丽隐杆线虫的化学遗传学研究发现,抗癌真菌毒素 Chaetocin 和 Chetomin 是核金属稳态反应的强效诱导剂

Abraham Elijah, Athapaththu A M Gihan K, Atanasova Kalina R, Chen Qi-Yin, Corcoran Taylor J, Piloto Juan, Wu Cheng-Wei, Ratnayake Ranjala, Luesch Hendrik, Choe Keith P

Isolation and Characterization of the Cyanobacterial Macrolide Glycoside Moorenaside, an Anti-Inflammatory Analogue of Aurisides Targeting the Keap1/Nrf2 Pathway

蓝藻大环内酯糖苷莫雷纳苷的分离与鉴定,莫雷纳苷是一种靶向Keap1/Nrf2通路的抗炎性Aurisides类似物

Al-Awadhi, Fatma H; Kokkaliari, Sofia; Ratnayake, Ranjala; Paul, Valerie J; Luesch, Hendrik

Discovery and Anti-Inflammatory Activity of a Cyanobacterial Fatty Acid Targeting the Keap1/Nrf2 Pathway

针对 Keap1/Nrf2 通路的蓝藻脂肪酸的发现及其抗炎活性

Fatma H Al-Awadhi, Emily F Simon, Na Liu, Ranjala Ratnayake, Valerie J Paul, Hendrik Luesch

Probing a distinct druggable tubulin binding site with gatorbulins 1-7, their metabolic and physicochemical properties, and pharmacological consequences

利用 gatorbulins 1-7 探测一种独特的、可成药的微管蛋白结合位点,研究其代谢和理化性质以及药理学后果

Qi-Yin Chen ,Ranjala Ratnayake ,Rafael Hortigüela ,Gustavo M Seabra ,Michael D Cameron ,J Fernando Díaz ,María Ángela Oliva ,Hendrik Luesch

Epigenetic Small-Molecule Screen for Inhibition and Reversal of Acinar Ductal Metaplasia in Mouse Pancreatic Organoids

利用表观遗传小分子筛选抑制和逆转小鼠胰腺类器官腺泡导管化生

Atanasova, Kalina R; Perkins, Corey M; Ratnayake, Ranjala; Jiang, Jinmai; Chen, Qi-Yin; Schmittgen, Thomas D; Luesch, Hendrik