日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Unbiased mapping of cereblon neosubstrate landscape by high-throughput proteomics.

利用高通量蛋白质组学对 cereblon 新底物景观进行无偏映射

Steger Martin, Nishiguchi Gisele, Wu Qiong, Schwalb Bjoern, Shashikadze Bachuki, McGowan Kevin, Actis Marisa, Aggarwal Anup, Shi Zhe, Price Jeanine, Mayasundari Anand, Yang Lei, Bednarz Anastasia H, Machata Sophie, Graef Tobias, Bartoschek Denis, Demichev Vadim, Ohmayer Uli, Yang Jun, Daub Henrik, Rankovic Zoran

ANGI-18. DISRUPTING INTEGRIN SIGNALING IMPAIRS MIGRATION, MYC-DRIVEN PURINE BIOSYNTHESIS, AND STEMNESS IN H3K27M DIFFUSE MIDLINE GLIOMAS

ANGI-18。干扰整合素信号传导会损害H3K27M弥漫性中线胶质瘤的迁移、MYC驱动的嘌呤生物合成和干性。

Angiolari, Federica; Coretti, Alessandro; Salanne, Mathieu; Bonella, Sara; Findlay, Izac; Staudt, Dilana; Duchatel, Ryan; Jackson, Evangeline; Persson, Mika; McEwen, Holly; Delevaux, Katherine; Smith, Nathan; Vitanza, Nicholas; Cain, Jason; Hansen, Mitchell; Alvaro, Frank; Jakobsen, Lene; Larsen, Martin; Savary, Clara; Waszak, Sebastian; Dun, Matthew; Ji, Sunjong; Doherty, Robert; Mota, Mateus; Natarajan, Siva Kumar; de la Nava, Daniel; Sajjakulnukit, Peter; Peterson, Erik R; Adam, Tiffany; Niculcea, Michael; Vo, Katie; Wink, Kelsey; Bavani, Subramaniam; Sridevi, Yadavilli; Nazarian, Javad; Phillips, Joanna J; Mueller, Sabine; Filbin, Mariella; Solomon, David A; Wahl, Daniel R; Lyssiotis, Costas; Qin, Tingting; Beck, Alexander; Viswanath, Pavithra; Nuechterlein, Nicholas; Waszak, Sebastian M; Venneti, Sriram; Koschmann, Carl; Schwark, Kallen; Miclea, Madeline; Patel, Tirth; Kong, Seongbae; Stanczak, Alina; Lau, Benison; Cartaxo, Rodrigo; Messinger, Dana; Doherty, Robert; Ji, Sunjong; Wadden, Jack; Clausen, Madison; Momen, Fareen; Adam, Tiffany; Wink, Kelsey; Hutchinson, Aria; Niculcea, Michael; Serhan, Habib; Merrill, Nathan; Edmonds, Amy; Mayr, Lisa; Neyazi, Sina; Muñoz, Denise; Nuechterlein, Nicholas; Fernandez, Ester Calvo; Califano, Andrea; Pavisic, Jovana; Garton, Hugh; Rao, Rama; Upadhyaya, Santhosh; Skrypek, Mary; Bendel, Anne; Lobbous, Mina; Klawinski, Darren; Merajver, Sofia; Koptyra, Mateusz; Resnick, Adam; Nazarian, Javad; Venneti, Sriram; Waszak, Sebastian; Chavez, Lukas; Beck, Alexander; Gojo, Johannes; Filbin, Mariella; Coppé, Jean-Philippe; Koschmann, Carl; Ahmad, Shiekh Tanveer; Li, Yiran; Garcia-Lopez, Jesus; Gudenas, Brian; Hadley, Jennifer; Paul, Leena; Wu, Stephanie; Refaat, Alaa; Kojic, Marija; Batts, Melissa; Soliman, Taha; Pitre, Aaron; Arnskötter, Frederik; Zindy, Frederique; Jones, Alun; Twarog, Nathaniel; Mayasundari, Anand; Bianski, Brandon; Tinkle, Christopher; Shirinifard, Abbas; Janke, Laura; Lu, Meifen; Lewis, Sara; Onar-Thomas, Arzu; Pfister, Stefan; Gajjar, Amar; Baker, Suzanne; Roussel, Martine; Rankovic, Zoran; Robinson, Giles; Orr, Brent; Wainwright, Brandon; Shelat, Anang; Waszak, Sebastian; Kutscher, Lena; Lin, Hong; Northcott, Paul; Doherty, Robert; Wink, Kelsey; Schwark, Kallen; Ji, Sunjong; Gera, Ananya; Messinger, Dana; de la Martin, Daniel Nava; Knowles, Truman; Subramaniam, Bavani; Millet, Yves; Waszak, Sebastian; Phillips, Joanna; Solomon, David; Nazarian, Javad; Mueller, Sabine; Beck, Alexander; Coppe, Jean-Phillipe; Koschmann, Carl; Cartaxo, Rodrigo T; de la Nava, Daniel; Nieblas-Bedolla, Edwin; Niculcea, Michael; Ji, Sunjong; Natarajan, Siva Kumar; Adam, Tiffany; Clausen, Madison; Miclea, Madeline; Siada, Ruby; Schwark, Kallen; Gera, Ananya; Doherty, Robert; Lyssiotis, Costas A; Favro, Noemi; Covato, Carmelo; Brunschwig, Lucas; Waszak, Sebastian M; Nuechterlein, Nicholas; Filbin, Mariella; Vo, Tuan; Dun, Matthew D; Venneti, Sriram; Hara, Toshiro; Koschmann, Carl

HTS Identifies NUP98-KDM5A-PHD3 Domain Ligands with Novel Scaffolds

高通量筛选鉴定出具有新型支架的NUP98-KDM5A-PHD3结构域配体

Lin, Wenwei; Slavish, P Jake; Phillips, Aaron H; Trotter, Marlon; Yang, Guangwei; Chai, Sergio C; Churion, Kelly; Ochoada, Jason; Das, Sourav; Shelat, Anang A; Mullighan, Charles G; Kriwacki, Richard W; Rankovic, Zoran; Chen, Taosheng

LCK-targeting molecular glues overcome resistance to inhibitor-based therapy in T-cell acute lymphoblastic leukemia

靶向LCK的分子胶克服了T细胞急性淋巴细胞白血病对抑制剂疗法的耐药性

Yang, Jun J; Nishiguchi, Gisele; Yoshimura, Satoshi; Actis, Marisa; Seffernick, Justin T; Jarusiewicz, Jamie A; Aggarwal, Anup; Li, Angelina; Li, Yong; Lee, DongGeun; Yang, Lei; Mayasundari, Anand; Rankovic, Zoran; Fischer, Marcus

Capmatinib is an effective treatment for MET-fusion driven pediatric high-grade glioma and synergizes with radiotherapy

卡马替尼是治疗MET融合基因驱动的儿童高级别胶质瘤的有效药物,并且与放射疗法具有协同作用。

Zuckermann, Marc; He, Chen; Andrews, Jared; Bagchi, Aditi; Sloan-Henry, Roketa; Bianski, Brandon; Xie, Jia; Wang, Yingzhe; Twarog, Nathaniel; Onar-Thomas, Arzu; Ernst, Kati J; Yang, Lei; Li, Yong; Zhu, Xiaoyan; Ocasio, Jennifer K; Budd, Kaitlin M; Dalton, James; Li, Xiaoyu; Chepyala, Divyabharathi; Zhang, Junyuan; Xu, Ke; Hover, Laura; Roach, Jordan T; Chan, Kenneth Chun-Ho; Hofmann, Nina; McKinnon, Peter J; Pfister, Stefan M; Shelat, Anang A; Rankovic, Zoran; Freeman, Burgess B 3rd; Chiang, Jason; Jones, David T W; Tinkle, Christopher L; Baker, Suzanne J

TMOD-19. GERMLINEELP1 DEFICIENCY SENSITIZES CEREBELLAR GRANULE NEURON PROGENITORS TO SHH MEDULLOBLASTOMA

TMOD-19. 生殖系ELP1缺陷使小脑颗粒神经元祖细胞对SHH髓母细胞瘤敏感

Schaufelberger, Luca; Blaskovits, J Terence; Laplaza, Ruben; Jorner, Kjell; Corminboeuf, Clemence; Kilburn, Lindsay; Franson, Andrea; Cooney, Tab; Kline, Cassie; Stoller, Schuyler; Reddy, Alyssa; Banerjee, Anu; Packer, Roger; Bendel, Anne; Skrypek, Maggie; Minturn, Jane; Abdelbaki, Mohamed; Whipple, Nicholas; Chan, Priya; Crawford, John; Crotty, Erin; Waanders, Angela; Elster, Jennifer; Raabe, Eric; George, Elizabeth; Pinto, Soniya; Supakul, Nucharin; Kraya, Adam; Prados, Michael; Nazarian, Javad; Solomon, David; Long-Boyle, Janel; Molinaro, Annette; Waszak, Sebastian; Mueller, Sabine; Tanveer Ahmad, Shiekh; Garcia-Lopez, Jesus; Li, Yiran; Hadley, Jennifer; Paul, Leena; Gudenas, Brian; Batts, Melissa; Soliman, Taha; Pitre, Aaron; Kojic, Marija; Manz, Frederik; Zindy, Frederique; Jones, Alun; Mayasundari, Anand; Bianski, Brandon; Tinkle, Christopher; Shirinifard, Abbas; Janke, Laura Janke; Lu, Meifen; Onar-Thomas, Arzu; Pfister, Stefan; Gajjar, Amar; Baker, Suzanne; Roussel, Martine; Rankovic, Zoran; Robinson, Giles; Orr, Brent; Wainwright, Brandon; Kutscher, Lena; Waszak, Sebastian; Lin, Hong; Northcott, Paul

Combination of Ribociclib with BET-Bromodomain and PI3K/mTOR Inhibitors for Medulloblastoma Treatment In Vitro and In Vivo

体外和体内研究Ribociclib联合BET-溴结构域抑制剂和PI3K/mTOR抑制剂治疗髓母细胞瘤

Jonchere, Barbara; Williams, Justin; Zindy, Frederique; Liu, Jingjing; Robinson, Sarah; Farmer, Dana M; Min, Jaeki; Yang, Lei; Stripay, Jennifer L; Wang, Yingzhe; Freeman, Burgess B; Yu, Jiyang; Shelat, Anang A; Rankovic, Zoran; Roussel, Martine F

Targeting KDM4 for treating PAX3-FOXO1-driven alveolar rhabdomyosarcoma

靶向KDM4治疗PAX3-FOXO1驱动的肺泡横纹肌肉瘤

Singh, Shivendra; Abu-Zaid, Ahmed; Jin, Hongjian; Fang, Jie; Wu, Qiong; Wang, Tingting; Feng, Helin; Quarni, Waise; Shao, Ying; Maxham, Lily; Abdolvahabi, Alireza; Yun, Mi-Kyung; Vaithiyalingam, Sivaraja; Tan, Haiyan; Bowling, John; Honnell, Victoria; Young, Brandon; Guo, Yian; Bajpai, Richa; Pruett-Miller, Shondra M; Grosveld, Gerard C; Hatley, Mark; Xu, Beisi; Fan, Yiping; Wu, Gang; Chen, Eleanor Y; Chen, Taosheng; Lewis, Peter W; Rankovic, Zoran; Li, Yimei; Murphy, Andrew J; Easton, John; Peng, Junmin; Chen, Xiang; Wang, Ruoning; White, Stephen W; Davidoff, Andrew M; Yang, Jun

Evaluating and evolving a screening library in academia: the St Jude approach

评估和发展学术界的筛查库:圣裘德儿童研究医院的方法

Nishiguchi, Gisele; Das, Sourav; Ochoada, Jason; Long, Heather; Lee, Richard E; Rankovic, Zoran; Shelat, Anang A

17-DMAG dually inhibits Hsp90 and histone lysine demethylases in alveolar rhabdomyosarcoma

17-DMAG 双重抑制肺泡横纹肌肉瘤中的 Hsp90 和组蛋白赖氨酸去甲基化酶

Singh, Shivendra; Abu-Zaid, Ahmed; Lin, Wenwei; Low, Jonathan; Abdolvahabi, Alireza; Jin, Hongjian; Wu, Qiong; Cooke, Bailey; Fang, Jie; Bowling, John; Vaithiyalingam, Sivaraja; Currier, Duane; Yun, Mi-Kyung; Fernando, Dinesh M; Maier, Julie; Tillman, Heather; Bulsara, Purva; Lu, Zhaohua; Das, Sourav; Shelat, Anang; Li, Zhenmei; Young, Brandon; Lee, Richard; Rankovic, Zoran; Murphy, Andrew J; White, Stephen W; Davidoff, Andrew M; Chen, Taosheng; Yang, Jun