日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Differentiating Inhibition Selectivity and Binding Affinity of Isocitrate Dehydrogenase 1 Variant Inhibitors

异柠檬酸脱氢酶 1 变体抑制剂的抑制选择性和结合亲和力的区分

Shuang Liu, Martine Abboud, Victor Mikhailov, Xiao Liu, Raphael Reinbold, Christopher J Schofield

Resistance to the isocitrate dehydrogenase 1 mutant inhibitor ivosidenib can be overcome by alternative dimer-interface binding inhibitors

异柠檬酸脱氢酶 1 突变抑制剂 ivosidenib 的耐药性可以通过替代二聚体界面结合抑制剂来克服

Raphael Reinbold, Ingvild C Hvinden #, Patrick Rabe #, Ryan A Herold, Alina Finch, James Wood, Melissa Morgan, Maximillian Staudt, Ian J Clifton, Fraser A Armstrong, James S O McCullagh, Jo Redmond, Chiara Bardella, Martine I Abboud, Christopher J Schofield