SAR Studies Leading to the Identification of a Novel Series of Metallo-β-lactamase Inhibitors for the Treatment of Carbapenem-Resistant Enterobacteriaceae Infections That Display Efficacy in an Animal Infection Model
SAR 研究鉴定出一系列新型金属β-内酰胺酶抑制剂,用于治疗耐碳青霉烯类肠杆菌感染,并在动物感染模型中显示出疗效。
期刊:ACS Infectious Diseases
影响因子:3.8
doi:10.1021/acsinfecdis.8b00246
Leiris, Simon; Coelho, Alicia; Castandet, Jérôme; Bayet, Maëlle; Lozano, Clarisse; Bougnon, Juliette; Bousquet, Justine; Everett, Martin; Lemonnier, Marc; Sprynski, Nicolas; Zalacain, Magdalena; Pallin, Thomas David; Cramp, Michael C; Jennings, Neil; Raphy, Gilles; Jones, Mark W; Pattipati, Ramesh; Shankar, Battu; Sivasubrahmanyam, Relangi; Soodhagani, Ashok K; Juventhala, Ramakrishna R; Pottabathini, Narender; Pothukanuri, Srinivasu; Benvenuti, Manuela; Pozzi, Cecilia; Mangani, Stefano; De Luca, Filomena; Cerboni, Giulia; Docquier, Jean-Denis; Davies, David T