Chemoprobe-based assays of histone lysine demethylase 1A target occupation enable in vivo pharmacokinetics and pharmacodynamics studies of KDM1A inhibitors
基于化学探针的组蛋白赖氨酸去甲基化酶 1A 靶标占据检测可用于进行 KDM1A 抑制剂的体内药代动力学和药效学研究
期刊:Journal of Biological Chemistry
影响因子:4
doi:10.1074/jbc.RA118.006980
Cristina Mascaró, Alberto Ortega, Elena Carceller, Raquel Ruiz Rodriguez, Filippo Ciceri, Serena Lunardi, Li Yu, Manuel Hilbert, Tamara Maes