日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Red Cell Distribution Width-Standard Deviation Is Associated with Cumulative Metabolic Burden but Not Independently with Metabolic Syndrome

红细胞分布宽度标准差与累积代谢负担相关,但与代谢综合征无独立相关性

Shereen; Tahir, Ayesha; Ahmed, Awais; Jan, Muhammad Saeed; Aslam, Nouman; Hassan, Sohail; Rashid, Umer; Lule, Kemal Ozan; Otay Lule, Nezihe; Savcilioglu, Mert Deniz; Yildiz, Hamit

Structure-Guided Design of Benzothiazole and Benzimidazole-Based Urea Derivatives Curtailing Oncogenic Signaling via Concurrent Inhibition of VEGFR-2, EGFR, and c‑Met

结构导向设计苯并噻唑和苯并咪唑类脲衍生物,通过同时抑制VEGFR-2、EGFR和c-Met来抑制致癌信号传导

Shaheen, Sadia; Siddique, Arshma; Iftikhar, Ali; Faisal, Amir; Rehman, Hafiz M; Murtaza, Ghulam; Tahir, Ayesha; Saeed, Anees; Hassan, Abbas; Rashid, Umer

Synthetic Derivates of Progesterone Ameliorate Scopolamine-Induced Cognitive Deficits in Animal Models: Antioxidant, Enzyme Inhibitory, Molecular Docking and Behavioral Correlates

合成孕酮衍生物可改善东莨菪碱诱导的动物模型认知缺陷:抗氧化、酶抑制、分子对接和行为相关性

Nawaz, Asif; Sadiq, Abdul; Bashir, Nasreena; Rashid, Umer; Ullah, Farhat; Khan, Shahbaz; Ullah, Farman; Khan, Mohammad Inam; Ayaz, Muhammad

Dihydropyrimidine-2-thione derivatives as SARS-CoV-2 main protease inhibitors: synthesis, SAR and in vitro profiling

二氢嘧啶-2-硫酮衍生物作为SARS-CoV-2主蛋白酶抑制剂:合成、构效关系及体外活性分析

Saeed, Anees; Tahir, Ayesha; Shah, Muhammad; Hussain, Fahad; Sadiq, Abdul; Rashid, Umer

Exploration of novel triazolo-thiadiazine hybrids of deferasirox as multi-target-directed anti-neuroinflammatory agents with structure-activity relationship (SAR): a new treatment opportunity for Alzheimer's disease.

探索新型三唑噻二嗪杂合物地拉罗司作为多靶点导向抗神经炎症药物的结构活性关系(SAR):阿尔茨海默病的新治疗机会

Shakir Syed Ahmed, Rashid Umer, Marryum, Fatima Nighat, Ejaz Syeda Abida, Fayyaz Ammara, Ullah Muhammad Zahid, Saeed Aamer, Khan Ajmal, Al Harrasi Ahmed, Mumtaz Amara

Correction: Mahnashi et al. In-Vitro, In-Vivo, Molecular Docking and ADMET Studies of 2-Substituted 3,7-Dihydroxy-4H-chromen-4-one for Oxidative Stress, Inflammation and Alzheimer's Disease. Metabolites 2022, 12, 1055

更正:Mahnashi 等人,《2-取代的 3,7-二羟基-4H-色烯-4-酮在氧化应激、炎症和阿尔茨海默病中的体外、体内、分子对接和 ADMET 研究》,《代谢物》2022, 12, 1055

Mahnashi, Mater H; Alshahrani, Mohammed Abdulrahman; Nahari, Mohammed H; Hassan, Syed Shams Ul; Jan, Muhammad Saeed; Ayaz, Muhammad; Ullah, Farhat; Alshehri, Osama M; Alshehri, Mohammad Ali; Rashid, Umer; Sadiq, Abdul

Anti-alkaline phosphatases (ALP) potentials of potent 4-aminobenzenesulfonamide derivatives against Naja oxiana venom

强效4-氨基苯磺酰胺衍生物对眼镜蛇毒液的抗碱性磷酸酶(ALP)活性

Khan, Saqib; Yaqoob, Muhammad; Asad, Muhammad H H B; Falak, Rafia; Ashraf, Zaman; Mannan, Abdul; Bukhari, Syed M; Alam, Fiaz; Rashid, Umer

Design, synthesis, and molecular docking studies of thiazole derivatives against phospholipase A(2) (Naja oxiana) venom

噻唑衍生物对抗磷脂酶A(2)(眼镜蛇)毒液的设计、合成和分子对接研究

Nayyab, Bibi F; Shah, Muhammad; Asad, Muhammad H H B; Zaidi, Asma; Alam, Fiaz; Mannan, Abdul; Rashid, Umer

Secondary metabolites isolated from Fernandoa adenophylla (Wall. ex G.Don) steenis as multitarget inhibitors of cholinesterases for the treatment of Alzheimer's Disease, followed by molecular docking studies.

从 Fernandoa adenophylla (Wall. ex G.Don) steenis 中分离出的次生代谢物作为胆碱酯酶的多靶点抑制剂用于治疗阿尔茨海默病,随后进行了分子对接研究

Maria, Khan Asifullah, Ajaj Rahaf, Rauf Abdur, Shah Zafar Ali, Ahmad Zubair, Hemeg Hassan A, Rashid Umer

Thymidine Phosphorylase Inhibitory Potential and Molecular Docking Studies of Secondary Metabolites Isolated From Fernandoa adenophylla (Wall. ex G. Don) Steenis

从腺叶费尔南多亚树(Fernandoa adenophylla (Wall. ex G. Don) Steenis)中分离的次生代谢产物的胸苷磷酸化酶抑制活性及分子对接研究

Rauf, Abdur; Khan, Majid; Rashid, Umer; Saeed, Anees; Shah, Zafar Ali; Ahmad, Zubair; Alamri, Abdulhakeem S; Alsanie, Walaa F; Khan, Imtiaz; Hussain, Humaira; Alhomrani, Majid; Iriti, Marcello