Rastelli Giulio相关文献与解析，生知库 | 链接生命科学的每一步

Citarella Andrea, Belluti Silvia, Bonanni Davide, Moi Davide, Piccinini Isabella, Rinaldi Arianna, Papulino Chiara, Benedetti Rosaria, Cuoghi Laura, Ciolo Stefano Di, Silvani Alessandra, Altucci Lucia, Pinzi Luca, Franchini Silvia, Passarella Daniele, Sorbi Claudia, Giannini Clelia, Imbriano Carol, Rastelli Giulio

肿瘤

前列腺癌

发表日期：2025

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Improving Machine Learning Classification Predictions through SHAP and Features Analysis Interpretation

通过SHAP和特征分析解释改进机器学习分类预测

期刊:Journal of Chemical Information and Modeling

影响因子:5.3

doi:10.1021/acs.jcim.5c02015

Bernal, Leonardo; Rastelli, Giulio; Pinzi, Luca

发表日期：2025

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Design, synthesis and biological activity of glycoconjugated ADAMTS5 exosite inhibitors: applications in osteoarthritis and ovarian cancer models.

糖缀合ADAMTS5外位点抑制剂的设计、合成和生物活性：在骨关节炎和卵巢癌模型中的应用。

期刊:Scientific Reports

影响因子:3.9

doi:10.1038/s41598-025-29549-3

Cuffaro Doretta, Blagg Sophie, Yamamoto Kazuhiro, Pinzi Luca, Bacchetti Rachele, Yuan Shengnan, Tew Simon, Campagnolo Paola, D'Andrea Felicia, Crispino Enrico, Rastelli Giulio, Rossello Armando, Rainero Elena, Nuti Elisa, Santamaria Salvatore

Early Diagnosis of Neurodegenerative Diseases: What Has Been Undertaken to Promote the Transition from PET to Fluorescence Tracers

神经退行性疾病的早期诊断：为促进从PET到荧光示踪剂的过渡已采取了哪些措施

期刊:Molecules

影响因子:4.6

doi:10.3390/molecules29030722

Bisi, Nicolò; Pinzi, Luca; Rastelli, Giulio; Tonali, Nicolò

神经科学

发表日期：2024

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Identification of Promising Drug Candidates against Prostate Cancer through Computationally-Driven Drug Repurposing

通过计算驱动的药物重定位来识别有前景的抗前列腺癌候选药物

期刊:International Journal of Molecular Sciences

影响因子:4.9

doi:10.3390/ijms24043135

Bernal, Leonardo; Pinzi, Luca; Rastelli, Giulio

Discovery of a Potent Dual Inhibitor of Aromatase and Aldosterone Synthase

发现一种强效的芳香化酶和醛固酮合成酶双重抑制剂

期刊:ACS Pharmacology and Translational Science

影响因子:3.7

doi:10.1021/acsptsci.3c00183

Tinivella, Annachiara; Banchi, Marta; Gambacorta, Guido; Borghi, Federica; Orlandi, Paola; Baxendale, Ian R; Di Paolo, Antonello; Bocci, Guido; Pinzi, Luca; Rastelli, Giulio

发表日期：2023

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Development of machine learning classifiers to predict compound activity on prostate cancer cell lines

开发机器学习分类器以预测化合物对前列腺癌细胞系的活性

期刊:Journal of Cheminformatics

影响因子:5.7

doi:10.1186/s13321-022-00647-y

Bonanni, Davide; Pinzi, Luca; Rastelli, Giulio

Identification of potential biological targets of oxindole scaffolds via in silico repositioning strategies

通过计算机模拟重定位策略鉴定吲哚骨架的潜在生物靶点

期刊:F1000Research

影响因子:

doi:10.12688/f1000research.109017.2

Tinivella, Annachiara; Pinzi, Luca; Gambacorta, Guido; Baxendale, Ian; Rastelli, Giulio

发表日期：2022

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LigAdvisor: a versatile and user-friendly web-platform for drug design

LigAdvisor：一个功能全面且用户友好的药物设计网络平台

期刊:Nucleic Acids Research

影响因子:13.1

doi:10.1093/nar/gkab385

Pinzi, Luca; Tinivella, Annachiara; Gagliardelli, Luca; Beneventano, Domenico; Rastelli, Giulio

发表日期：2021

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Hydroxamic Acid Derivatives: From Synthetic Strategies to Medicinal Chemistry Applications

羟肟酸衍生物：从合成策略到药物化学应用

期刊:ACS Omega

影响因子:4.3

doi:10.1021/acsomega.1c03628

Citarella, Andrea; Moi, Davide; Pinzi, Luca; Bonanni, Davide; Rastelli, Giulio

发表日期：2021

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Structure-Based Discovery of Hsp90/HDAC6 Dual Inhibitors Targeting Aggressive Prostate Cancer.

基于结构的Hsp90/HDAC6双重抑制剂的发现及其在侵袭性前列腺癌中的应用

Improving Machine Learning Classification Predictions through SHAP and Features Analysis Interpretation

通过SHAP和特征分析解释改进机器学习分类预测

Design, synthesis and biological activity of glycoconjugated ADAMTS5 exosite inhibitors: applications in osteoarthritis and ovarian cancer models.

糖缀合ADAMTS5外位点抑制剂的设计、合成和生物活性：在骨关节炎和卵巢癌模型中的应用。

Early Diagnosis of Neurodegenerative Diseases: What Has Been Undertaken to Promote the Transition from PET to Fluorescence Tracers

神经退行性疾病的早期诊断：为促进从PET到荧光示踪剂的过渡已采取了哪些措施

Identification of Promising Drug Candidates against Prostate Cancer through Computationally-Driven Drug Repurposing

通过计算驱动的药物重定位来识别有前景的抗前列腺癌候选药物

Discovery of a Potent Dual Inhibitor of Aromatase and Aldosterone Synthase

发现一种强效的芳香化酶和醛固酮合成酶双重抑制剂

Development of machine learning classifiers to predict compound activity on prostate cancer cell lines

开发机器学习分类器以预测化合物对前列腺癌细胞系的活性

Identification of potential biological targets of oxindole scaffolds via in silico repositioning strategies

通过计算机模拟重定位策略鉴定吲哚骨架的潜在生物靶点

LigAdvisor: a versatile and user-friendly web-platform for drug design

LigAdvisor：一个功能全面且用户友好的药物设计网络平台

Hydroxamic Acid Derivatives: From Synthetic Strategies to Medicinal Chemistry Applications

羟肟酸衍生物：从合成策略到药物化学应用