日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Design, Synthesis, and Biological Evaluation of Novel Acetylcholinesterase and β-Secretase 1 Inhibitors

新型乙酰胆碱酯酶和β-分泌酶1抑制剂的设计、合成及生物学评价

Drozdowska, Danuta; Pawelski, Damian; Wróbel-Tałałaj, Agnieszka; Plonska-Brzezinska, Marta; Kolesinska, Beata; Lazny, Ryszard; Seroka, Barbara; Parzych, Cezary; Ratkiewicz, Artur

Substituent and Ring-Number Effects on the Kinetics of PAH + OH Reactions: A QSAR-DOE Approach with Tunneling Corrections

取代基和环数对PAH + OH反应动力学的影响:基于隧道效应校正的QSAR-DOE方法

Parzych, Cezary; Baradyn, Maciej; Ratkiewicz, Artur

Rational design, synthesis, and molecular modelling insights of dual DNA binders/DHFR inhibitors bearing arylidene-hydrazinyl-1,3-thiazole scaffold with apoptotic and anti-migratory potential in breast MCF-7 cancer cells.

对具有亚芳基肼基-1,3-噻唑骨架的双重DNA结合剂/DHFR抑制剂进行合理设计、合成和分子建模,以研究其在乳腺癌MCF-7细胞中的凋亡和抗迁移潜力

El-Wakil Marwa H, Ghazala Rasha A, El-Dershaby Hadeel A, Drozdowska Danuta, Wróbel-Tałałaj Agnieszka, Parzych Cezary, Ratkiewicz Artur, Kolesińska Beata, Abd El-Razik Heba A, Soliman Farid S G

Repurposed Arylidene-hydrazinyl-1,3-thiazoles as Multitarget Anti-Alzheimer's Agents via Combined Computational and Experimental Studies

通过计算和实验相结合的研究,将亚芳基肼基-1,3-噻唑类化合物重新用于多靶点抗阿尔茨海默病治疗

Drozdowska, Danuta; Ratkiewicz, Artur; Wróbel-Tałałaj, Agnieszka; Parzych, Cezary; El-Dershaby, Hadeel A; Abd El-Razik, Heba A; Soliman, Farid S G; El-Wakil, Marwa H

A highly variable habitat selection in moose across diel and seasonal scales

驼鹿的栖息地选择在昼夜和季节尺度上具有高度可变性

Borowik, Tomasz; Kowalczyk, Rafał; Ratkiewicz, Mirosław; Maślanko, Weronika; Duda, Norbert; Żmihorski, Michał

Benzamide Trimethoprim Derivatives as Human Dihydrofolate Reductase Inhibitors-Molecular Modeling and In Vitro Activity Study

苯甲酰胺类甲氧苄啶衍生物作为人二氢叶酸还原酶抑制剂——分子建模和体外活性研究

Drozdowska, Danuta; Wróbel-Tałałaj, Agnieszka; Parzych, Cezary; Ratkiewicz, Artur

In Vitro and In Silico Studies on Cytotoxic Properties of Oxythiamine and 2'-Methylthiamine

氧硫胺和 2'-甲硫胺的细胞毒特性的体外和计算机模拟研究

Marta Malinowska, Magdalena Czerniecka, Izabella Jastrzebska, Artur Ratkiewicz, Adam Tylicki, Natalia Wawrusiewicz-Kurylonek

New Steroidal Selenides as Proapoptotic Factors

新型甾体硒化物作为促凋亡因子

Izabella Jastrzebska, Natalia Wawrusiewicz-Kurylonek, Paweł A Grześ, Artur Ratkiewicz, Ewa Grabowska, Magdalena Czerniecka, Urszula Czyżewska, Adam Tylicki

Tail feather strength in tail-assisted climbing birds is achieved through geometric, not material change

尾羽强度在尾部辅助攀爬的鸟类中是通过几何形状的变化而非材料的变化来实现的。

Dickinson, Edwin; Young, Melody W; DeLeon, David; Bas, Burcak; Zou, Bettina; Ratkiewicz, Aleksandra; Beatty, Brian L; Granatosky, Michael C

Genome-environment association analyses reveal geographically restricted adaptive divergence across the range of the widespread Eurasian carnivore Lynx lynx (Linnaeus, 1758)

基因组-环境关联分析揭示了广泛分布于欧亚大陆的食肉动物猞猁(Lynx lynx (Linnaeus, 1758))在其分布范围内存在地理限制的适应性分化。

Bazzicalupo, Enrico; Ratkiewicz, Mirosław; Seryodkin, Ivan V; Okhlopkov, Innokentiy; Galsandorj, Naranbaatar; Yarovenko, Yuriy A; Ozolins, Janis; Saveljev, Alexander P; Melovski, Dime; Gavashelishvili, Alexander; Schmidt, Krzysztof; Godoy, José A