日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Correction: Progress in the discovery and development of anticancer agents from marine cyanobacteria

更正:海洋蓝藻抗癌药物的发现和开发进展

Luesch, Hendrik; Ellis, Emma K; Chen, Qi-Yin; Ratnayake, Ranjala

Progress in the discovery and development of anticancer agents from marine cyanobacteria

海洋蓝藻抗癌药物的发现与开发进展

Luesch, Hendrik; Ellis, Emma K; Chen, Qi-Yin; Ratnayake, Ranjala

Morphological profiling for drug discovery in the era of deep learning

深度学习时代药物发现的形态学分析

Tang, Qiaosi; Ratnayake, Ranjala; Seabra, Gustavo; Jiang, Zhe; Fang, Ruogu; Cui, Lina; Ding, Yousong; Kahveci, Tamer; Bian, Jiang; Li, Chenglong; Luesch, Hendrik; Li, Yanjun

Biosynthesis of Dolastatin 10 in Marine Cyanobacteria, a Prototype for Multiple Approved Cancer Drugs

海洋蓝藻中多拉司他汀10的生物合成,是多种已获批准的抗癌药物的原型

Kallifidas, Dimitris; Dhakal, Dipesh; Chen, Manyun; Chen, Qi-Yin; Kokkaliari, Sofia; Colon Rosa, Nicole A; Ratnayake, Ranjala; Bruner, Steven D; Paul, Valerie J; Ding, Yousong; Luesch, Hendrik

Chemical Genetics in C. elegans Identifies Anticancer Mycotoxins Chaetocin and Chetomin as Potent Inducers of a Nuclear Metal Homeostasis Response.

秀丽隐杆线虫的化学遗传学研究发现,抗癌真菌毒素 Chaetocin 和 Chetomin 是核金属稳态反应的强效诱导剂

Abraham Elijah, Athapaththu A M Gihan K, Atanasova Kalina R, Chen Qi-Yin, Corcoran Taylor J, Piloto Juan, Wu Cheng-Wei, Ratnayake Ranjala, Luesch Hendrik, Choe Keith P

Isolation and Characterization of the Cyanobacterial Macrolide Glycoside Moorenaside, an Anti-Inflammatory Analogue of Aurisides Targeting the Keap1/Nrf2 Pathway

蓝藻大环内酯糖苷莫雷纳苷的分离与鉴定,莫雷纳苷是一种靶向Keap1/Nrf2通路的抗炎性Aurisides类似物

Al-Awadhi, Fatma H; Kokkaliari, Sofia; Ratnayake, Ranjala; Paul, Valerie J; Luesch, Hendrik

Epigenetic Small-Molecule Screen for Inhibition and Reversal of Acinar Ductal Metaplasia in Mouse Pancreatic Organoids

利用表观遗传小分子筛选抑制和逆转小鼠胰腺类器官腺泡导管化生

Atanasova, Kalina R; Perkins, Corey M; Ratnayake, Ranjala; Jiang, Jinmai; Chen, Qi-Yin; Schmittgen, Thomas D; Luesch, Hendrik

Gatorbulin-1, a distinct cyclodepsipeptide chemotype, targets a seventh tubulin pharmacological site

Gatorbulin-1 是一种独特的环状缩肽化学类型,靶向第七个微管蛋白药理学位点。

Matthew, Susan; Chen, Qi-Yin; Ratnayake, Ranjala; Fermaintt, Charles S; Lucena-Agell, Daniel; Bonato, Francesca; Prota, Andrea E; Lim, Seok Ting; Wang, Xiaomeng; Díaz, J Fernando; Risinger, April L; Paul, Valerie J; Oliva, Maria Ángela; Luesch, Hendrik

Seaweed natural products modify the host inflammatory response via Nrf2 signaling and alter colon microbiota composition and gene expression.

海藻天然产物通过 Nrf2 信号通路调节宿主的炎症反应,并改变结肠微生物群组成和基因表达

Bousquet Michelle S, Ratnayake Ranjala, Pope Jillian L, Chen Qi-Yin, Zhu Fanchao, Chen Sixue, Carney Thomas J, Gharaibeh Raad Z, Jobin Christian, Paul Valerie J, Luesch Hendrik

Largazole is a Brain-Penetrant Class I HDAC Inhibitor with Extended Applicability to Glioblastoma and CNS Diseases

Largazole是一种可穿透血脑屏障的I类HDAC抑制剂,具有广泛的应用前景,可用于治疗胶质母细胞瘤和中枢神经系统疾病。

Al-Awadhi, Fatma H; Salvador-Reyes, Lilibeth A; Elsadek, Lobna A; Ratnayake, Ranjala; Chen, Qi-Yin; Luesch, Hendrik