日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Discovery of First-in-Class Carbonic Anhydrase/Histone Deacetylase Dual Inhibitors with Antiproliferative Activity in Cancer Cells

发现具有抗癌细胞增殖活性的首创碳酸酐酶/组蛋白去乙酰化酶双重抑制剂

Bozdag, Murat; Mroweh, Nabil; Raucci, Alessia; Angeli, Andrea; Peppicelli, Silvia; Biagioni, Alessio; Calorini, Lido; Trisciuoglio, Daniela; Ragno, Rino; Astolfi, Roberta; Giuliani, Lidia; Zwergel, Clemens; Valente, Sergio; Andreucci, Elena; Carta, Fabrizio; Mai, Antonello; Supuran, Claudiu T

Advancements in Hydrazide-Based HDAC Inhibitors: A Review of Recent Developments and Therapeutic Potential

基于酰肼的HDAC抑制剂的研究进展:近期进展及治疗潜力综述

Raucci, Alessia; Zwergel, Clemens; Valente, Sergio; Mai, Antonello

Quinoline-Based DNA Methyltransferase Inhibitors Featuring Basic Side Chains: Design, Synthesis, and Insight in Biochemical and Anticancer Cell Properties

具有碱性侧链的喹啉类DNA甲基转移酶抑制剂:设计、合成及其生化和抗癌细胞特性研究

Zwergel, Clemens; Lambona, Chiara; Fioravanti, Rossella; Raucci, Alessia; Fiorentino, Francesco; Nchugoua Tchieh, Guilaine; Jallet, Corinne; Lacroix, Laurent; Pierrettori, Michela; Pellegrini, Francesca Romana; Xiong, Yan; Jin, Jian; Arimondo, Paola; Trisciuoglio, Daniela; Mai, Antonello; Valente, Sergio

Procognitive Potential of Neuroprotective Triazine 5-HT(6) Receptor Antagonists Tested on Chronic Activity In Vivo in Rats: Computer-Aided Insight into the Role of Chalcogen-Differences on the Pharmacological Profile.

在大鼠体内慢性活动中测试神经保护性三嗪 5-HT(6) 受体拮抗剂的促认知潜力:计算机辅助深入了解硫族元素差异对药理学特征的作用

Jastrzębska-Więsek Magdalena, Garbo Sabrina, Cios Agnieszka, Wilczyńska-Zawal Natalia, Partyka Anna, Honkisz-Orzechowska Ewelina, Å»esławska Ewa, Handzlik Jarosław, Mordyl Barbara, Głuch-Lutwin Monika, Raucci Alessia, Hittinger Marius, Starek Małgorzata, DÄ browska Monika, Nitek Wojciech, Karcz Tadeusz, Skórkowska Alicja, Gdula-Argasińska Joanna, Czarnota-Łydka Kinga, Pyka Patryk, Szymańska Ewa, Kucwaj-Brysz Katarzyna, Zwergel Clemens, Wesołowska Anna, Battistelli Cecilia, Handzlik Jadwiga