日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Lipid Pocket Binders Impose Allosteric Changes of Protein Dynamics Around the Active Site of the Protein Kinase p38α

脂质口袋结合物引起蛋白激酶p38α活性位点周围蛋白质动力学的变构变化

Medina Gómez, Sara; Homberg, Laurin T; Bührmann, Mike; Rauh, Daniel; Linser, Rasmus

Elimusertib enhances cytotoxic effects of conventional chemotherapy and sensitizes to radiation in preclinical Ewing sarcoma models

Elimusertib可增强传统化疗的细胞毒性作用,并在临床前尤文氏肉瘤模型中提高放射治疗的敏感性。

Koch, Leonhard; Kerkhoff, Maximilian; Bretschneider, Maximilian; Dayi, Samet; Plaumann, Pauline; Sadeghi, Bahareh; Maaßen, Emma; Hillesheim, Emilia; Kuballa, Marc; Schaefer, Christiane; Rauh, Daniel; Grunewald, Susanne; Bauer, Sebastian; von Neubeck, Cläre; Dirksen, Uta

Computational Design of Lysine Targeting Covalent Binders Using Rosetta.

利用 Rosetta 进行赖氨酸靶向共价结合剂的计算设计

Tivon Barr, Wiese Jan, Müller Matthias P, Gabizon Ronen, Rauh Daniel, London Nir

Advancing TET Inhibitor Development: From Structural Insights to Biological Evaluation

推进TET抑制剂的研发:从结构解析到生物学评价

Willems, Suzanne; Maksumic, Lejla; Niggenaber, Janina; Lin, Tzu-Chen; Schulz, Tom; Weisner, Jörn; Sievers, Sonja; Müller, Matthias P; Summerer, Daniel; Rauh, Daniel

Targeting KRAS(G13C) with cyclic linker based inhibitors to explore warhead orientation

利用基于环状连接子的抑制剂靶向KRAS(G13C)以探索弹头取向

Kirschner, Tonia; Rodriguez, João; Moreira, Emerson Gonçalves; Niggenaber, Janina; Warmuth, Jonas D; Verli, Hugo; Müller, Matthias P; Rauh, Daniel

KIT ATP-Binding Pocket/Activation Loop Mutations in GI Stromal Tumor: Emerging Mechanisms of Kinase Inhibitor Escape

胃肠道间质瘤中KIT ATP结合口袋/激活环突变:激酶抑制剂逃逸的新机制

Mühlenberg, Thomas; Falkenhorst, Johanna; Schulz, Tom; Fletcher, Benjamin S; Teuber, Alina; Krzeciesa, Dawid; Klooster, Isabella; Lundberg, Meijun; Wilson, Lydia; Lategahn, Jonas; von Mehren, Margaret; Grunewald, Susanne; Tüns, Alicia Isabell; Wardelmann, Eva; Sicklick, Jason K; Brahmi, Mehdi; Serrano, César; Schildhaus, Hans-Ulrich; Sievers, Sonja; Treckmann, Jürgen; Heinrich, Michael C; Raut, Chandrajit P; Ou, Wen-Bin; Marino-Enriquez, Adrian; George, Suzanne; Rauh, Daniel; Fletcher, Jonathan A; Bauer, Sebastian

Design and synthesis of Nrf2-derived hydrocarbon stapled peptides for the disruption of protein-DNA-interactions.

设计和合成 Nrf2 衍生的碳氢化合物交联肽,以破坏蛋白质-DNA 相互作用

Wiedemann Bianca, Kamps Dominic, Depta Laura, Weisner Jörn, Cvetreznik Jana, Tomassi Stefano, Gentz Sascha, Hoffmann Jan-Erik, Müller Matthias P, Koch Oliver, Dehmelt Leif, Rauh Daniel

KRasG12C inhibitors in clinical trials: a short historical perspective

KRasG12C抑制剂的临床试验:简要历史回顾

Goebel, Lisa; Müller, Matthias P; Goody, Roger S; Rauh, Daniel

Covalent-Allosteric Inhibitors to Achieve Akt Isoform-Selectivity

共价变构抑制剂实现Akt亚型选择性

Quambusch, Lena; Landel, Ina; Depta, Laura; Weisner, Jörn; Uhlenbrock, Niklas; Müller, Matthias P; Glanemann, Franziska; Althoff, Kristina; Siveke, Jens T; Rauh, Daniel

Donated chemical probes for open science

捐赠化学探针用于开放科学

Müller, Susanne; Ackloo, Suzanne; Arrowsmith, Cheryl H; Bauser, Marcus; Baryza, Jeremy L; Blagg, Julian; Böttcher, Jark; Bountra, Chas; Brown, Peter J; Bunnage, Mark E; Carter, Adrian J; Damerell, David; Dötsch, Volker; Drewry, David H; Edwards, Aled M; Edwards, James; Elkins, Jon M; Fischer, Christian; Frye, Stephen V; Gollner, Andreas; Grimshaw, Charles E; IJzerman, Adriaan; Hanke, Thomas; Hartung, Ingo V; Hitchcock, Steve; Howe, Trevor; Hughes, Terry V; Laufer, Stefan; Li, Volkhart Mj; Liras, Spiros; Marsden, Brian D; Matsui, Hisanori; Mathias, John; O'Hagan, Ronan C; Owen, Dafydd R; Pande, Vineet; Rauh, Daniel; Rosenberg, Saul H; Roth, Bryan L; Schneider, Natalie S; Scholten, Cora; Singh Saikatendu, Kumar; Simeonov, Anton; Takizawa, Masayuki; Tse, Chris; Thompson, Paul R; Treiber, Daniel K; Viana, Amélia Yi; Wells, Carrow I; Willson, Timothy M; Zuercher, William J; Knapp, Stefan; Mueller-Fahrnow, Anke