日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Novel Deazaflavin Analogues Potently Inhibited Tyrosyl DNA Phosphodiesterase 2 (TDP2) and Strongly Sensitized Cancer Cells toward Treatment with Topoisomerase II (TOP2) Poison Etoposide

新型脱氮黄素类似物可有效抑制酪氨酰DNA磷酸二酯酶2 (TDP2),并显著增强癌细胞对拓扑异构酶II (TOP2) 抑制剂依托泊苷的敏感性。

Kankanala, Jayakanth; Ribeiro, Carlos J A; Kiselev, Evgeny; Ravji, Azhar; Williams, Jessica; Xie, Jiashu; Aihara, Hideki; Pommier, Yves; Wang, Zhengqiang

New fluorescence-based high-throughput screening assay for small molecule inhibitors of tyrosyl-DNA phosphodiesterase 2 (TDP2)

一种基于荧光的新型高通量筛选酪氨酰-DNA磷酸二酯酶2(TDP2)小分子抑制剂的方法

Ribeiro, Carlos J A; Kankanala, Jayakanth; Shi, Ke; Kurahashi, Kayo; Kiselev, Evgeny; Ravji, Azhar; Pommier, Yves; Aihara, Hideki; Wang, Zhengqiang

Synthesis and Biological Evaluation of the First Triple Inhibitors of Human Topoisomerase 1, Tyrosyl-DNA Phosphodiesterase 1 (Tdp1), and Tyrosyl-DNA Phosphodiesterase 2 (Tdp2).

人类拓扑异构酶 1、酪氨酰-DNA 磷酸二酯酶 1 (Tdp1) 和酪氨酰-DNA 磷酸二酯酶 2 (Tdp2) 的首个三重抑制剂的合成和生物学评价

Wang Ping, Elsayed Mohamed S A, Plescia Caroline B, Ravji Azhar, Redon Christophe E, Kiselev Evgeny, Marchand Christophe, Zeleznik Olga, Agama Keli, Pommier Yves, Cushman Mark