Synthesis and Biological Evaluation of the First Triple Inhibitors of Human Topoisomerase 1, Tyrosyl-DNA Phosphodiesterase 1 (Tdp1), and Tyrosyl-DNA Phosphodiesterase 2 (Tdp2).
人类拓扑异构酶 1、酪氨酰-DNA 磷酸二酯酶 1 (Tdp1) 和酪氨酰-DNA 磷酸二酯酶 2 (Tdp2) 的首个三重抑制剂的合成和生物学评价
期刊:Journal of Medicinal Chemistry
影响因子:6.8
doi:10.1021/acs.jmedchem.6b01565
Wang Ping, Elsayed Mohamed S A, Plescia Caroline B, Ravji Azhar, Redon Christophe E, Kiselev Evgeny, Marchand Christophe, Zeleznik Olga, Agama Keli, Pommier Yves, Cushman Mark