日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Multi-targeted azacoumarin-cyanocinnamate hybrids induce G(2)/M arrest and apoptosis via tubulin, and COX-2/VEGFR modulation: insights from in vitro mechanistic basis and in vivo validation

多靶点氮杂香豆素-氰基肉桂酸酯杂合物通过微管蛋白和COX-2/VEGFR调控诱导G2/M期阻滞和细胞凋亡:来自体外机制基础和体内验证的见解

El-Zend, Manar A; El-Deen, Ibrahim M; Mansour, Rawda M; Yousef, Tarek A; Alrashidi, Amal Abdullah; Saied, Essa M

Discovery of benzochromene derivatives first example with dual cytotoxic activity against the resistant cancer cell MCF-7/ADR and inhibitory effect of the P-glycoprotein expression levels

发现苯并色烯衍生物首例对耐药癌细胞MCF-7/ADR具有双重细胞毒活性及抑制P-糖蛋白表达水平的作用

Lali M Al-Harbi, Eman A Al-Harbi, Rawda M Okasha, R A El-Eisawy, Mohammed A A El-Nassag, Hany M Mohamed, Ahmed M Fouda, Ahmed A Elhenawy, Ahmed Mora, Ahmed M El-Agrody, Heba K A El-Mawgoud

Synthesis and Characterization of a New Class of Chromene-Azo Sulfonamide Hybrids as Promising Anticancer Candidates with the Exploration of Their EGFR, h CAII, and MMP-2 Inhibitors Based on Molecular Docking Assays

基于分子对接分析,合成和表征一类新型色满-偶氮磺酰胺杂化物,作为有前途的抗癌候选药物,并探索其对 EGFR、h CAII 和 MMP-2 的抑制剂作用

Fawzia F Alblewi, Mosa H Alsehli, Zainab M Hritani, Areej Eskandrani, Wael H Alsaedi, Majed O Alawad, Ahmed A Elhenawy, Hanaa Y Ahmed, Mohamed S A El-Gaby, Tarek H Afifi, Rawda M Okasha

Core shell stationary phase for a novel separation of some COVID-19 used drugs by UPLC-MS/MS Method: Study of grapefruit consumption impact on their pharmacokinetics in rats

采用核壳固定相通过 UPLC-MS/MS 方法分离部分 COVID-19 所用药物:研究食用葡萄柚对大鼠体内药代动力学的影响

Sally Tarek Mahmoud, Marwa A Moffid, Rawda M Sayed, Eman A Mostafa

Novel 2-Hydroselenonicotinonitriles and Selenopheno[2, 3-b]pyridines: Efficient Synthesis, Molecular Docking-DFT Modeling, and Antimicrobial Assessment

新型2-氢硒烟腈和硒吩并[2,3-b]吡啶:高效合成、分子对接-DFT建模及抗菌活性评价

Abdellattif, Magda H; Abdel-Rahman, Adel A H; Arief, Mohamed Mohamed Helmy; Mouneir, Samar M; Ali, Amena; Hussien, Mostafa A; Okasha, Rawda M; Afifi, Tarek H; Hagar, Mohamed

A New Family of Benzo[ h]Chromene Based Azo Dye: Synthesis, In-Silico and DFT Studies with In Vitro Antimicrobial and Antiproliferative Assessment

一类新的苯并[h]色烯基偶氮染料:合成、计算机模拟和 DFT 研究以及体外抗菌和抗增殖评估

Alaa S Abd-El-Aziz, Azhaar Alsaggaf, Eman Assirey, Arshi Naqvi, Rawda M Okasha, Tarek H Afifi, Mohamed Hagar

Synthesis, Biological Assessment, and Structure Activity Relationship Studies of New Flavanones Embodying Chromene Moieties

含色烯部分的新型黄烷酮的合成、生物评价及构效关系研究

Eman Assirey, Azhaar Alsaggaf, Arshi Naqvi, Ziad Moussa, Rawda M Okasha, Tarek H Afifi, Alaa S Abd-El-Aziz

Design of Novel Oligomeric Mixed Ligand Complexes: Preparation, Biological Applications and the First Example of Their Nanosized Scale

新型低聚混合配体复合物的设计:制备、生物学应用及其纳米尺度的首例研究

Okasha, Rawda M; Al-Shaikh, Najla E; Aljohani, Faizah S; Naqvi, Arshi; Ismail, Eman H

Rational Design and Synthesis of Diverse Pyrimidine Molecules Bearing Sulfonamide Moiety as Novel ERK Inhibitors

合理设计和合成含有磺酰胺部分的多种嘧啶分子作为新型 ERK 抑制剂

Ahmed H Halawa, Areej A Eskandrani, Walid E Elgammal, Saber M Hassan, Ahmed H Hassan, Hassan Y Ebrahim, Ahmed B M Mehany, Ahmed M El-Agrody, Rawda M Okasha

Introducing novel potent anticancer agents of 1H-benzo[f]chromene scaffolds, targeting c-Src kinase enzyme with MDA-MB-231 cell line anti-invasion effect

介绍 1H-苯并[f]色烯骨架的新型强效抗癌剂,靶向 c-Src 激酶,具有 MDA-MB-231 细胞系抗侵袭作用

Hany E A Ahmed, Mohammed A A El-Nassag, Ahmed H Hassan, Rawda M Okasha, Saleh Ihmaid, Ahmed M Fouda, Tarek H Afifi, Ateyatallah Aljuhani, Ahmed M El-Agrody