日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Exploring Integrin α5β1 as a Potential Therapeutic Target for Pulmonary Arterial Hypertension: Insights From Comprehensive Multicenter Preclinical Studies

探索整合素α5β1作为肺动脉高压潜在治疗靶点:来自综合多中心临床前研究的启示

Lemay, Sarah-Eve; Montesinos, Mónica S; Grobs, Yann; Yokokawa, Tetsuro; Shimauchi, Tsukasa; Mougin, Manon; Romanet, Charlotte; Sauvaget, Mélanie; Breuils-Bonnet, Sandra; Bourgeois, Alice; Théberge, Charlie; Pelletier, Andréanne; El Kabbout, Reem; Martineau, Sandra; Yamamoto, Keiko; Akram, Muzaffar; Ray, Adrian S; Lippa, Blaise; Goodwin, Bryan; Lin, Fu-Yang; Wang, Hua; Dowling, James E; Lu, Min; Qiao, Qi; McTeague, T Andrew; Moy, Terence I; Potus, François; Provencher, Steeve; Boucherat, Olivier; Bonnet, Sébastien

Acetyl-CoA Carboxylase Inhibition Reverses NAFLD and Hepatic Insulin Resistance but Promotes Hypertriglyceridemia in Rodents

乙酰辅酶A羧化酶抑制剂可逆转非酒精性脂肪性肝病和肝脏胰岛素抵抗,但会促进啮齿动物高甘油三酯血症。

Goedeke, Leigh; Bates, Jamie; Vatner, Daniel F; Perry, Rachel J; Wang, Ting; Ramirez, Ricardo; Li, Li; Ellis, Matthew W; Zhang, Dongyan; Wong, Kari E; Beysen, Carine; Cline, Gary W; Ray, Adrian S; Shulman, Gerald I

Transporters in Drug Development: 2018 ITC Recommendations for Transporters of Emerging Clinical Importance

药物研发中的转运体:2018 年 ITC 关于新兴临床重要转运体的建议

Zamek-Gliszczynski, Maciej J; Taub, Mitchell E; Chothe, Paresh P; Chu, Xiaoyan; Giacomini, Kathleen M; Kim, Richard B; Ray, Adrian S; Stocker, Sophie L; Unadkat, Jashvant D; Wittwer, Matthias B; Xia, Cindy; Yee, Sook-Wah; Zhang, Lei; Zhang, Yan

Nucleotide Prodrug Containing a Nonproteinogenic Amino Acid To Improve Oral Delivery of a Hepatitis C Virus Treatment

含有非蛋白源性氨基酸的核苷酸前药可改善丙型肝炎病毒治疗药物的口服递送

Feng, Joy Y; Wang, Ting; Park, Yeojin; Babusis, Darius; Birkus, Gabriel; Xu, Yili; Voitenleitner, Christian; Fenaux, Martijn; Yang, Huiling; Eng, Stacey; Tirunagari, Neeraj; Kirschberg, Thorsten; Cho, Aesop; Ray, Adrian S

Sofosbuvir and Ribavirin Liver Pharmacokinetics in Patients Infected with Hepatitis C Virus

丙型肝炎病毒感染患者体内索非布韦和利巴韦林的肝脏药代动力学

Babusis, Darius; Curry, Michael P; Kirby, Brian; Park, Yeojin; Murakami, Eisuke; Wang, Ting; Mathias, Anita; Afdhal, Nezam; McHutchison, John G; Ray, Adrian S

Transporter Expression in Noncancerous and Cancerous Liver Tissue from Donors with Hepatocellular Carcinoma and Chronic Hepatitis C Infection Quantified by LC-MS/MS Proteomics

利用液相色谱-串联质谱蛋白质组学定量分析肝细胞癌和慢性丙型肝炎感染供体非癌性和癌性肝组织中转运蛋白的表达

Billington, Sarah; Ray, Adrian S; Salphati, Laurent; Xiao, Guangqing; Chu, Xiaoyan; Humphreys, W Griffith; Liao, Mingxiang; Lee, Caroline A; Mathias, Anita; Hop, Cornelis E C A; Rowbottom, Christopher; Evers, Raymond; Lai, Yurong; Kelly, Edward J; Prasad, Bhagwat; Unadkat, Jashvant D

Broad-spectrum antiviral GS-5734 inhibits both epidemic and zoonotic coronaviruses

广谱抗病毒药物GS-5734可抑制流行性冠状病毒和人畜共患冠状病毒。

Sheahan, Timothy P; Sims, Amy C; Graham, Rachel L; Menachery, Vineet D; Gralinski, Lisa E; Case, James B; Leist, Sarah R; Pyrc, Krzysztof; Feng, Joy Y; Trantcheva, Iva; Bannister, Roy; Park, Yeojin; Babusis, Darius; Clarke, Michael O; Mackman, Richard L; Spahn, Jamie E; Palmiotti, Christopher A; Siegel, Dustin; Ray, Adrian S; Cihlar, Tomas; Jordan, Robert; Denison, Mark R; Baric, Ralph S

Role of Mitochondrial Toxicity in BMS-986094-Induced Toxicity

线粒体毒性在BMS-986094诱导毒性中的作用

Feng, Joy Y; Tay, Chin H; Ray, Adrian S

Transporter Expression in Liver Tissue from Subjects with Alcoholic or Hepatitis C Cirrhosis Quantified by Targeted Quantitative Proteomics

利用靶向定量蛋白质组学方法定量分析酒精性肝硬化或丙型肝炎肝硬化患者肝组织中转运蛋白的表达

Wang, Li; Collins, Carol; Kelly, Edward J; Chu, Xiaoyan; Ray, Adrian S; Salphati, Laurent; Xiao, Guangqing; Lee, Caroline; Lai, Yurong; Liao, Mingxiang; Mathias, Anita; Evers, Raymond; Humphreys, William; Hop, Cornelis E C A; Kumer, Sean C; Unadkat, Jashvant D

Implications of efficient hepatic delivery by tenofovir alafenamide (GS-7340) for hepatitis B virus therapy

替诺福韦艾拉酚胺(GS-7340)高效肝脏递送对乙型肝炎病毒治疗的意义

Murakami, Eisuke; Wang, Ting; Park, Yeojin; Hao, Jia; Lepist, Eve-Irene; Babusis, Darius; Ray, Adrian S