日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Structural and dynamic features of cagrilintide binding to calcitonin and amylin receptors.

卡格里林肽与降钙素和胰淀素受体结合的结构和动力学特征

Cao Jianjun, Belousoff Matthew J, Johnson Rachel M, Keov Peter, Mariam Zamara, Deganutti Giuseppe, Christopoulos George, Hick Caroline A, Reedtz-Runge Steffen, Glendorf Tine, Ballarín-González Borja, Raun Kirsten, Bayly-Jones Charles, Wootten Denise, Sexton Patrick M

A GLP-1 analogue optimized for cAMP-biased signaling improves weight loss in obese mice.

针对 cAMP 偏向信号传导优化的 GLP-1 类似物可改善肥胖小鼠的体重减轻

Douros Jonathan D, Novikoff Aaron, DuBois Barent, Rohlfs Rebecca, Mokrosinski Jacek, Hogendorf Wouter F J, Augustin Robert, Merkestein Myrte, Egaa Martini Lene Brandt, Linderoth Lars, Gerrard Elliot, Kodra Janos Tibor, Norlin Jenny, Roed Nikolaj Kulahin, Oldenburger Anouk, Mowery Stephanie A, Waldhoer Maria, Perez-Tilve Diego, Finan Brian, Reedtz-Runge Steffen, Müller Timo D, Knerr Patrick J

Full-length human GLP-1 receptor structure without orthosteric ligands

不含正位配体的全长人GLP-1受体结构

Wu, Fan; Yang, Linlin; Hang, Kaini; Laursen, Mette; Wu, Lijie; Han, Gye Won; Ren, Qiansheng; Roed, Nikolaj Kulahin; Lin, Guangyao; Hanson, Michael A; Jiang, Hualiang; Wang, Ming-Wei; Reedtz-Runge, Steffen; Song, Gaojie; Stevens, Raymond C

Structural insight into antibody-mediated antagonism of the Glucagon-like peptide-1 Receptor

抗体介导的胰高血糖素样肽-1受体拮抗作用的结构解析

Hennen, Stephanie; Kodra, János T; Soroka, Vladyslav; Krogh, Berit O; Wu, Xiaoai; Kaastrup, Peter; Ørskov, Cathrine; Rønn, Sif G; Schluckebier, Gerd; Barbateskovic, Silvia; Gandhi, Prafull S; Reedtz-Runge, Steffen

Structural Determinants of Binding the Seven-transmembrane Domain of the Glucagon-like Peptide-1 Receptor (GLP-1R)

胰高血糖素样肽-1受体(GLP-1R)七次跨膜结构域结合的结构决定因素

Yang, Dehua; de Graaf, Chris; Yang, Linlin; Song, Gaojie; Dai, Antao; Cai, Xiaoqing; Feng, Yang; Reedtz-Runge, Steffen; Hanson, Michael A; Yang, Huaiyu; Jiang, Hualiang; Stevens, Raymond C; Wang, Ming-Wei