日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Structure-Guided Design of a KMT9 Inhibitor Prodrug with Cellular Activity.

基于结构的KMT9抑制剂前药设计及其细胞活性

Wang Sheng, Barthes Nicolas P F, Urban Sylvia, Hazai Viktor I, Klein Sebastian O, Pappert Tabea, Kümmel Paul, Heller Nicolas, Bacher Johannes, Staudt Maximilian, Ruprecht Jan, Peng Ling, Sum Manuela, Berlin Christopher, Sarraf Daad, Regenass Pierre, Warstat Robin, Walz Johannes, Mishra Pankaj, Zhang Lin, Einsle Oliver, Günther Stefan, Breit Bernhard, Metzger Eric, Jung Manfred, Schüle Roland

The bactericidal FabI inhibitor Debio 1453 clears antibiotic-resistant Neisseria gonorrhoeae infection in vivo

杀菌性FabI抑制剂Debio 1453可在体内清除耐抗生素的淋病奈瑟菌感染。

Gerusz, Vincent; Regenass, Pierre; Rousseau, Quentin; Moraine, Victor; Dao, Justine; Lavé, Xavier; Das, Shampa; Hue Perron, Josée; Fajas Descamps, Laurence; Bravo, Juan; Dieppois, Guennaëlle; Kaplan, Nachum; Lefebre, Matthew; Altomari, Deanna; Romanov, Vladimir; Finn, Terry; Daram, Pierre; Bernardini, Francesca; Gross, Michaël; Lysek, Robert; Adam, Aurélien; Pohin, Danig; Maio, Maurizio; Tatsis, Vasileios; Sunose, Mihiro; Ronin, Céline; Ciesielski, Fabrice; Ahlstrand, Josefine; Jacobsson, Susanne; Unemo, Magnus; Cameron, David R

Structure-Based Design, Docking and Binding Free Energy Calculations of A366 Derivatives as Spindlin1 Inhibitors

基于结构的A366衍生物作为Spindlin1抑制剂的设计、对接和结合自由能计算

Luise, Chiara; Robaa, Dina; Regenass, Pierre; Maurer, David; Ostrovskyi, Dmytro; Seifert, Ludwig; Bacher, Johannes; Burgahn, Teresa; Wagner, Tobias; Seitz, Johannes; Greschik, Holger; Park, Kwang-Su; Xiong, Yan; Jin, Jian; Schüle, Roland; Breit, Bernhard; Jung, Manfred; Sippl, Wolfgang