日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Host- and pathogen-related determinants of pulmonary versus extrapulmonary tuberculosis

肺结核与肺外结核的宿主和病原体相关决定因素

Tulu, Begna; Brehm, Thomas Theo; van Crevel, Reinout; Dallenga, Tobias; DiNardo, Andrew R; Dheda, Keertan; Eggeling, Johanna; Enbiale, Wendemagegn; Gröschel, Matthias I; Hao, Jialun; Kumar, Vinod; van Laarhoven, Arjan; Londt, Rolanda; Prosser, Gareth; Randall, Philippa; Reiling, Norbert; Rybniker, Jan; Schaible, Ulrich E; Schurr, Erwin; Suarez, Isabelle; Theobald, Sebastian J; Wilkinson, Robert J; Lange, Christoph

Identification of Natural-Product Inhibitors of the 2C‑Methyl‑d‑erythritol 4‑Phosphate Pathway

2C-甲基-D-赤藓糖醇4-磷酸途径天然产物抑制剂的鉴定

Diamanti, Eleonora; Alhayek, Alaa; Lacour, Antoine; Shahrour, Mohammad Walid; Willocx, Daan; Illarionov, Boris; Fischer, Markus; Stadler, Marc; Reiling, Norbert; Herrmann, Jennifer; Müller, Rolf; Hirsch, Anna K H

Design and optimization of simplified inhibitors targeting Escherichia coli and Klebsiella pneumoniae IspE

设计和优化针对大肠杆菌和肺炎克雷伯菌 IspE 的简化抑制剂

Walsh, Danica J; Hamid, Rawia; Giele, Tim; Reiling, Norbert; Rottmann, Matthias; Hamed, Mostafa M; Hirsch, Anna K H

Positive Charge in an Antimalarial Compound Unlocks Broad-Spectrum Antibacterial Activity

抗疟化合物中的正电荷可释放广谱抗菌活性

Braun-Cornejo, Maria; Platteschorre, Mitchell; de Vries, Vincent; Bravo, Patricia; Sonawane, Vidhisha; Hamed, Mostafa M; Haupenthal, Jörg; Reiling, Norbert; Rottmann, Matthias; Piet, Dennis; Maas, Peter; Diamanti, Eleonora; Hirsch, Anna K H

Engineering an Artificial Myxopyronin Derivative with Enhanced Metabolic Stability via Mutasynthesis

通过突变合成工程构建具有增强代谢稳定性的人工粘液吡喃酮衍生物

Kiefer, Alexander F; Voltz, Alexander; Scherzer, Domen; Reberšek, Roman; Kany, Andreas M; Prosser, Gareth; Neuber, Markus; Reiling, Norbert; Hirsch, Anna K H; Müller, Rolf

Design, Synthesis, and Biological Evaluation of Mono- and Diamino-Substituted Squaramide Derivatives as Potent Inhibitors of Mycobacterial Adenosine Triphosphate (ATP) Synthase

单氨基和二氨基取代的方酰胺衍生物作为结核分枝杆菌腺苷三磷酸(ATP)合成酶的强效抑制剂的设计、合成和生物学评价

Palme, Paul R; Grover, Shipra; Abdelaziz, Rana; Mann, Lea; Kany, Andreas M; Ouologuem, Lina; Bartel, Karin; Sonnenkalb, Lindsay; Reiling, Norbert; Hirsch, Anna K H; Schnappinger, Dirk; Rubinstein, John L; Imming, Peter; Richter, Adrian

SMAD2 linker phosphorylation impacts overall survival, proliferation, TGFβ1-dependent gene expression and pluripotency-related proteins in NSCLC.

SMAD2 连接子磷酸化影响非小细胞肺癌的总体生存率、增殖、TGFβ1 依赖性基因表达和多能性相关蛋白

Nitschkowski Dörte, Vierbuchen Tim, Heine Holger, Behrends Jochen, Reiling Norbert, Reck Martin, Rabe Klaus F, Kugler Christian, Ammerpohl Ole, Drömann Daniel, Muley Thomas, Kriegsmann Mark, Stathopoulos Georgious T, Arendt Kristina A M, Goldmann Torsten, Marwitz Sebastian

Synthesis and Antimycobacterial Assays of Some New Ethambutol Analogs

合成及抗结核分枝杆菌活性测定:几种新型乙胺丁醇类似物

Abdelaziz, Rana; Dube, Mthandazo; Mann, Lea; Richter, Adrian; Robaa, Dina; Reiling, Norbert; Abdel-Halim, Mohammad; Imming, Peter

GlnA3(Mt) is able to glutamylate spermine but it is not essential for the detoxification of spermine in Mycobacterium tuberculosis

GlnA3(Mt)能够谷氨酰化亚精胺,但它并非结核分枝杆菌中亚精胺解毒所必需。

Krysenko, Sergii; Emani, Carine Sao; Bäuerle, Moritz; Oswald, Maria; Kulik, Andreas; Meyners, Christian; Hillemann, Doris; Merker, Matthias; Prosser, Gareth; Wohlers, Inken; Hausch, Felix; Brötz-Oesterhelt, Heike; Mitulski, Agnieszka; Reiling, Norbert; Wohlleben, Wolfgang

Spermine enhances the activity of anti-tuberculosis drugs

精胺能增强抗结核药物的活性

Sao Emani, Carine; Reiling, Norbert