Synthesis of a potent and selective (18)F-labeled delta-opioid receptor antagonist derived from the Dmt-Tic pharmacophore for positron emission tomography imaging
合成一种高效且选择性的(18)F标记δ-阿片受体拮抗剂,该拮抗剂源自Dmt-Tic药效团,用于正电子发射断层扫描成像
期刊:Journal of Medicinal Chemistry
影响因子:6.8
doi:10.1021/jm7014765
Ryu, Eun Kyoung; Wu, Zhanhong; Chen, Kai; Lazarus, Lawrence H; Marczak, Ewa D; Sasaki, Yusuke; Ambo, Akihiro; Salvadori, Severo; Ren, Chuancheng; Zhao, Heng; Balboni, Gianfranco; Chen, Xiaoyuan