日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

A STING agonist prodrug reprograms tumor-associated macrophage to boost colorectal cancer immunotherapy

一种STING激动剂前药可重编程肿瘤相关巨噬细胞,从而增强结直肠癌免疫疗法。

Aohua Deng ,Renming Fan ,Yongrui Hai ,Junyan Zhuang ,Bingjie Zhang ,Xintong Lu ,Wenhui Wang ,Li Luo ,Ge Bai ,Lei Liang ,Le Yang ,Minggao Zhao ,Gaofei Wei

An immunometabolic prodrug strategy overcomes DHODH inhibitor resistance in refractory melanoma

免疫代谢前药策略克服了难治性黑色素瘤中DHODH抑制剂的耐药性

Yongrui Hai # ,Wenhui Wang # ,Renming Fan # ,Ye Chen # ,Junyan Zhuang ,Shuo Fu ,Guiquan Ding ,Lei Liang ,Junke Song ,Gaofei Wei

Novel Pt(IV) complex OAP2 induces STING activation and pyroptosis via mitochondrial membrane remodeling for synergistic chemo-immunotherapy

新型Pt(IV)配合物OAP2通过线粒体膜重塑诱导STING激活和细胞焦亡,从而实现化疗-免疫疗法的协同作用。

Renming Fan ,Ruizhuo Lin ,Shuo Zhang ,Aohua Deng ,Yongrui Hai ,Junyan Zhuang ,Yang Liu ,Maosheng Cheng ,Gaofei Wei

A novel mitochondria-targeting DHODH inhibitor induces robust ferroptosis and alleviates immune suppression

一种新型的线粒体靶向 DHODH 抑制剂可诱导强烈的铁死亡并减轻免疫抑制

Yongrui Hai, Renming Fan, Ting Zhao, Ruizhuo Lin, Junyan Zhuang, Aohua Deng, Shanshui Meng, Zhuang Hou, Gaofei Wei

A platinum(IV)-artesunate complex triggers ferroptosis by boosting cytoplasmic and mitochondrial lipid peroxidation to enhance tumor immunotherapy

铂(IV)-青蒿琥酯复合物通过促进细胞质和线粒体脂质过氧化引发铁死亡,从而增强肿瘤免疫治疗

Renming Fan, Aohua Deng, Ruizhuo Lin, Shuo Zhang, Caiyan Cheng, Junyan Zhuang, Yongrui Hai, Minggao Zhao, Le Yang, Gaofei Wei

CJ2: A Novel Potent Platinum(IV) Prodrug Enhances Chemo-Immunotherapy by Facilitating PD-L1 Degradation in the Cytoplasm and Cytomembrane

CJ2:一种新型强效铂(IV)前药,通过促进细胞质和细胞膜中的 PD-L1 降解来增强化学免疫疗法

Renming Fan, Aohua Deng, Bing Qi, Shuo Zhang, Ruoxi Sang, Lanxin Luo, Jiakui Gou, Yongqing Liu, Ruizhuo Lin, Minggao Zhao, Yang Liu, Le Yang, Maosheng Cheng, Gaofei Wei