日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Antiprotozoal dimeric naphthylisoquinolines, mbandakamines B3 and B4, and related 5,8'-coupled monomeric alkaloids, ikelacongolines A-D, from a Congolese Ancistrocladus liana

抗原虫二聚萘异喹啉、mbandakamines B3 和 B4,以及相关的 5,8'-偶联单体生物碱、ikelacongolines AD,来自刚果 Ancistrocladus liana

Jean-Pierre Mufusama, Doris Feineis, Virima Mudogo, Marcel Kaiser, Reto Brun, Gerhard Bringmann

Synthesis of novel amide and urea derivatives of thiazol-2-ethylamines and their activity against Trypanosoma brucei rhodesiense

噻唑-2-乙胺新型酰胺和脲衍生物的合成及其对罗得西亚锥虫的活性

Donald A Patrick ,Tanja Wenzler ,Sihyung Yang ,Patrick T Weiser ,Michael Zhuo Wang ,Reto Brun ,Richard R Tidwell

Alkanediamide-Linked Bisbenzamidines Are Promising Antiparasitic Agents

烷二酰胺连接的双苯甲脒是一种很有前途的抗寄生虫药物

Jean J Vanden Eynde, Annie Mayence, Madhusoodanan Mottamal, Cyrus J Bacchi, Nigel Yarlett, Marcel Kaiser, Reto Brun, Tien L Huang

Evaluation of the in vitro trypanocidal activity of methylated flavonoid constituents of Vitex simplicifolia leaves

评价单叶荆条叶甲基化黄酮类成分的体外杀锥虫活性

Ngozi Nwodo, Festus Okoye, Daowan Lai, Abdesammed Debbab, Marcel Kaiser, Reto Brun, Peter Proksch

Two trypanocidal dipeptides from the roots of Zapoteca portoricensis (Fabaceae)

豆科植物 Zapoteca portoricensis 根中的两种锥虫二肽

Ngozi Justina Nwodo, Festus Basden C Okoye, Daowan Lai, Abdessamad Debbab, Reto Brun, Peter Proksch

UV-triggered affinity capture identifies interactions between the Plasmodium falciparum multidrug resistance protein 1 (PfMDR1) and antimalarial agents in live parasitized cells

紫外线触发的亲和力捕获可识别活寄生细胞中恶性疟原虫多药耐药蛋白 1 (PfMDR1) 与抗疟药物之间的相互作用

Ralf Brunner, Caroline L Ng, Hamed Aissaoui, Myles H Akabas, Christoph Boss, Reto Brun, Paul S Callaghan, Olivier Corminboeuf, David A Fidock, Ithiel J Frame, Bibia Heidmann, Amélie Le Bihan, Paul Jenö, Corinna Mattheis, Suzette Moes, Ingrid B Müller, Michelle Paguio, Paul D Roepe, Romain Siegrist, 

Anti-protozoal activity of aporphine and protoberberine alkaloids from Annickia kummeriae (Engl. & Diels) Setten & Maas (Annonaceae)

番荔枝科 (Annickia kummeriae) (Engl. & Diels) Setten & Maas 的阿朴啡和原小檗碱的抗原虫活性

Hamisi M Malebo, Tanja Wenzler, Monical Cal, Sauda M Swaleh, Maurice O Omolo, Ahmed Hassanali, Urs Séquin, Daniel Häussinger, Petur Dalsgaard, Matthias Hamburger, Reto Brun, Isaiah O Ndiege

Genetic reconstruction of protozoan rRNA decoding sites provides a rationale for paromomycin activity against Leishmania and Trypanosoma

原生动物 rRNA 解码位点的遗传重建为巴龙霉素对抗利什曼原虫和锥虫的活性提供了理论依据

Sven N Hobbie, Marcel Kaiser, Sebastian Schmidt, Dmitri Shcherbakov, Tanja Janusic, Reto Brun, Erik C Böttger

Synthesis, structure-activity relationship, and mode-of-action studies of antimalarial reversed chloroquine compounds

抗疟逆转氯喹化合物的合成、构效关系及作用方式研究

Steven J Burgess, Jane X Kelly, Shawheen Shomloo, Sergio Wittlin, Reto Brun, Katherine Liebmann, David H Peyton

Trypanothione reductase high-throughput screening campaign identifies novel classes of inhibitors with antiparasitic activity

锥虫硫酮还原酶高通量筛选活动确定了具有抗寄生虫活性的新型抑制剂

Georgina A Holloway, William N Charman, Alan H Fairlamb, Reto Brun, Marcel Kaiser, Edmund Kostewicz, Patrizia M Novello, John P Parisot, John Richardson, Ian P Street, Keith G Watson, Jonathan B Baell