Development and Characterization of pFluor50, a Fluorogenic-Based Kinetic Assay System for High-Throughput Inhibition Screening and Characterization of Time-Dependent Inhibition and Inhibition Type for Six Human CYPs.
pFluor50 的开发和表征,一种基于荧光的动力学分析系统,用于高通量抑制筛选和表征六种人类 CYP 的时间依赖性抑制和抑制类型
期刊:Molecules
影响因子:4.6
doi:10.3390/molecules30092032
Shriwas Pratik, Revnew Andre, Roo Sarah, Bender Alex, Miller Kevin, Hadad Christopher M, Lane Thomas R, Ekins Sean, McElroy Craig A