日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Evaluation of the antitumor activity of NOV202, a novel microtubule targeting and vascular disrupting agent

新型微管靶向和血管破坏剂 NOV202 的抗肿瘤活性评估

Linda Rickardson, Emma Kutvonen, Satu Orasniemi, Marita Högberg, Marko J Kallio, Stefan Rehnmark

Drug screen in patient cells suggests quinacrine to be repositioned for treatment of acute myeloid leukemia

患者细胞药物筛选表明,奎宁有望用于治疗急性髓系白血病。

Eriksson, A; Österroos, A; Hassan, S; Gullbo, J; Rickardson, L; Jarvius, M; Nygren, P; Fryknäs, M; Höglund, M; Larsson, R

Induction of mitochondrial dysfunction as a strategy for targeting tumour cells in metabolically compromised microenvironments

诱导线粒体功能障碍作为在代谢受损的微环境中靶向肿瘤细胞的一种策略

Xiaonan Zhang, Mårten Fryknäs, Emma Hernlund, Walid Fayad, Angelo De Milito, Maria Hägg Olofsson, Vladimir Gogvadze, Long Dang, Sven Påhlman, Leoni A Kunz Schughart, Linda Rickardson, Padraig D'Arcy, Joachim Gullbo, Peter Nygren, Rolf Larsson, Stig Linder

Screening for phenotype selective activity in multidrug resistant cells identifies a novel tubulin active agent insensitive to common forms of cancer drug resistance

通过对多药耐药细胞中的表型选择性活性进行筛选,可鉴定出一种对常见形式的癌症耐药性不敏感的新型微管蛋白活性剂

Mårten Fryknäs, Joachim Gullbo, Xin Wang, Linda Rickardson, Malin Jarvius, Malin Wickström, Saadia Hassan, Claes Andersson, Mats Gustafsson, Gunnar Westman, Peter Nygren, Stig Linder, Rolf Larsson

Stat1 activation attenuates IL-6 induced Stat3 activity but does not alter apoptosis sensitivity in multiple myeloma

Stat1 激活可减弱 IL-6 诱导的 Stat3 活性,但不会改变多发性骨髓瘤的细胞凋亡敏感性

Lina Y Dimberg, Anna Dimberg, Karolina Ivarsson, Mårten Fryknäs, Linda Rickardson, Gerard Tobin, Simon Ekman, Rolf Larsson, Urban Gullberg, Kenneth Nilsson, Fredrik Öberg, Helena Jernberg Wiklund

High content screening for inhibitors of protein interactions and post-translational modifications in primary cells by proximity ligation

通过邻位连接高内涵筛选原代细胞中蛋白质相互作用和翻译后修饰的抑制剂

Karl-Johan Leuchowius, Malin Jarvius, Malin Wickström, Linda Rickardson, Ulf Landegren, Rolf Larsson, Ola Söderberg, Mårten Fryknäs, Jonas Jarvius